TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Competitive antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of CAP-induced intracellular Ca2+ influx prein...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataKd: 0.589nMAssay Description:Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKd: 0.0640nMAssay Description:Binding affinity to rat TRPV1 after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Displacement of [3H]A-778317 from human TRPV1 expressed in CHO cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataKd: 0.590nMAssay Description:Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair