Affinity DataKd: 0.5nM EC50: 1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataKd: 588nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 0.5nM EC50: 1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataKd: 61nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 5.90nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 1.85E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
Affinity DataKd: 1.85E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
Affinity DataKd: 629nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+4nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 2.10nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 588nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.126nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.251nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 158nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.398nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Binding affinity to DOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Binding affinity to DOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 625nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 910nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 715nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 1.98E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 1.98E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 0.25 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 0.25 nM concentration expressed as dissociation consta...More data for this Ligand-Target Pair
Affinity DataKd: 4.30nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2.30nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+4nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 0.450nM EC50: 1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair