Compile Data Set for Download or QSAR
maximum 50k data
Found 47 of kd data for polymerid = 2100,3138,49000863,49000865
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKd:  0.5nM EC50:  1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021322(3-(3-Methyl-1-phenethyl-piperidin-3-yl)-phenol | 3...)
Affinity DataKd:  588nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKd:  0.5nM EC50:  1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001551(22-cyclopropylmethyl-9-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  61nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001553(22-cyclopropylmethyl-8-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  5.60nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001552(22-cyclopropylmethyl-7-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  5.90nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001554(22-cyclopropylmethyl-6-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  15nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKd:  1.85E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKd:  1.85E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataKd:  629nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021327(3-(1,3-Dimethyl-piperidin-3-yl)-phenol | 3-(1,3-Di...)
Affinity DataKd:  3.00E+4nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50452273(Dihydromorphine)
Affinity DataKd:  100nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKd:  2.10nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021323(3-(1-Allyl-3-methyl-piperidin-3-yl)-phenol | 3-(1-...)
Affinity DataKd:  4.00E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021322(3-(3-Methyl-1-phenethyl-piperidin-3-yl)-phenol | 3...)
Affinity DataKd:  588nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060064(2-[(R)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  2.5nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060065(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  0.126nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060082(2-({2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-met...)
Affinity DataKd:  0.251nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060072(2-[(R)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  158nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060076(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  2.5nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060068(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  0.398nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060075(2-({2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKd:  1.60nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50060071(2-[(S)-3-(4-Hydroxy-2,6-dimethyl-phenyl)-2-methyla...)
Affinity DataKd:  3.20nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM50037134((+)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKd:  20nMAssay Description:Binding affinity to human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to DOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM50346951(CHEMBL1795711 | CHEMBL1795714)
Affinity DataKd:  0.240nMAssay Description:Binding affinity to DOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKd:  18nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021324(3-(1-Cyclopropylmethyl-3-methyl-piperidin-3-yl)-ph...)
Affinity DataKd:  2.70E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021328(3-Cyclopropylmethyl-11-ethyl-8-hydroxy-6-methyl-3,...)
Affinity DataKd:  14nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019093(1-Cyclopropylmethyl-3-(3-hydroxy-phenyl)-piperidin...)
Affinity DataKd:  260nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019097(1-Cyclopropylmethyl-3-(3-hydroxy-phenyl)-2-methyl-...)
Affinity DataKd:  625nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019095(1-Allyl-3-(3-hydroxy-phenyl)-2-methyl-piperidine-3...)
Affinity DataKd:  770nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019098(3-(3-Hydroxy-phenyl)-1,2-dimethyl-piperidine-3-car...)
Affinity DataKd:  910nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019091(3-(3-Hydroxy-phenyl)-2-methyl-1-phenethyl-piperidi...)
Affinity DataKd:  170nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019092(3-(3-Hydroxy-phenyl)-1-methyl-piperidine-3-carboxy...)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019094(1-Allyl-3-(3-hydroxy-phenyl)-piperidine-3-carboxyl...)
Affinity DataKd:  715nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKd:  1.98E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKd:  1.98E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001553(22-cyclopropylmethyl-8-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  40nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 0.25 nM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001552(22-cyclopropylmethyl-7-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  37nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 0.25 nM concentration expressed as dissociation consta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001554(22-cyclopropylmethyl-6-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  4.30nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001551(22-cyclopropylmethyl-9-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  16nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001551(22-cyclopropylmethyl-9-isothiocyanato-14-oxa-11,22...)
Affinity DataKd:  2.30nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021327(3-(1,3-Dimethyl-piperidin-3-yl)-phenol | 3-(1,3-Di...)
Affinity DataKd:  3.00E+4nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021324(3-(1-Cyclopropylmethyl-3-methyl-piperidin-3-yl)-ph...)
Affinity DataKd:  2.70E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021323(3-(1-Allyl-3-methyl-piperidin-3-yl)-phenol | 3-(1-...)
Affinity DataKd:  4.00E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKd:  0.450nM EC50:  1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed