Affinity DataKd: 1.30nM EC50: 27nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataKd: 0.25nMAssay Description:The equilibrium binding constant to guinea pig cerebral cortex membranes was measuredMore data for this Ligand-Target Pair
Affinity DataKd: 8.10nMAssay Description:The equilibrium binding constant to pig cerebral cortex membranes was measuredMore data for this Ligand-Target Pair
Affinity DataKd: 0.110nMAssay Description:The equilibrium binding constant to guinea pig cerebral cortex membranes was measuredMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Tested in vitro for gastrin binding to gastrin receptors from guinea pig gastric glandsMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
Affinity DataKd: 22nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKd: 1.40nMAssay Description:Tested in vitro by the gastrin binding assay for the competitive binding with iodinated gastrin for the gastrin receptors in AR42J cellsMore data for this Ligand-Target Pair