Compile Data Set for Download or QSAR
Report error Found 309 of kd data for polymerid = 2888,5366,49000244,49000246,50002775,50007095
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404791BDBM50404791(CHEMBL31025)
Affinity DataKd:  0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404774BDBM50404774(CHEMBL31857)
Affinity DataKd:  0.00000100nMAssay Description:In vivo inhibition of Beta-1 adrenergic receptor in guinea pig right atria after 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404790BDBM50404790(CHEMBL13284)
Affinity DataKd:  0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404790BDBM50404790(CHEMBL13284)
Affinity DataKd:  0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404793BDBM50404793(CHEMBL31638)
Affinity DataKd:  0.0000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404763BDBM50404763(CHEMBL283289)
Affinity DataKd:  0.0000100nMAssay Description:In vivo inhibition of Beta-1 adrenergic receptor in guinea pig right atria after 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404796BDBM50404796(Brevibloc | ESMOLOL)
Affinity DataKd:  0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404796BDBM50404796(Brevibloc | ESMOLOL)
Affinity DataKd:  0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404804BDBM50404804(CHEMBL13365)
Affinity DataKd:  0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50568740BDBM50568740(CHEMBL4860528)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50601567BDBM50601567(CHEMBL5206565)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50601551BDBM50601551(CHEMBL5207281)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50601574BDBM50601574(CHEMBL5201074)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404789BDBM50404789(CHEMBL30622)
Affinity DataKd:  0.100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25746BDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25748BDBM25748(ICI 89,406 | 3-(2-{[3-(2-cyanophenoxy)-2-hydroxypr...)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292219BDBM50292219((2S)-1-(tert-butylamino)-3-[(4-morpholin-4-yl-1,2,...)
Affinity DataKd:  0.363nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241366BDBM50241366((S)-1-(isopropylamino)-3-(m-tolyloxy)propan-2-ol (...)
Affinity DataKd:  0.380nMAssay Description:Binding affinity to beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25747BDBM25747(4-[3-(tert-butylamino)-2-hydroxypropoxy]-2,3-dihyd...)
Affinity DataKd:  0.620nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2008
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404980BDBM50404980(CHEMBL1788320)
Affinity DataKd:  0.851nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404978BDBM50404978(CHEMBL173424)
Affinity DataKd:  0.851nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404987BDBM50404987(CHEMBL3085291)
Affinity DataKd:  0.891nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232757BDBM50232757(CHEMBL4092412)
Affinity DataKd:  0.977nMAssay Description:Displacement of [3H](-)CGP12177 from human beta1-AR expressed in CHOK1 cells after 2 hrs by TopCount microscintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432704BDBM50432704(CHEMBL2348218)
Affinity DataKd:  1nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25746BDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H](-)CGP12177 from human beta1-AR expressed in CHOK1 cells after 2 hrs by TopCount microscintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404988BDBM50404988(CHEMBL11171)
Affinity DataKd:  1.20nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25748BDBM25748(ICI 89,406 | 3-(2-{[3-(2-cyanophenoxy)-2-hydroxypr...)
Affinity DataKd:  1.24nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2008
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432701BDBM50432701(CHEMBL2348201)
Affinity DataKd:  1.5nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404804BDBM50404804(CHEMBL13365)
Affinity DataKd:  1.60nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404982BDBM50404982(CHEMBL366769)
Affinity DataKd:  1.60nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25746BDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKd:  1.60nMAssay Description:Displacement of [3H]-CGP12177 from human beta1 adrenoceptor expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25746BDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKd:  1.60nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2008
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432707BDBM50432707(LK-204-545 | LK-204545)
Affinity DataKd:  1.70nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405521BDBM50405521(ALO 1401-02 | ALO-1401-02 | Betaxolol | BETAXOLOL ...)
Affinity DataKd:  1.70nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKd:  1.70nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25759BDBM25759([3-(9H-carbazol-4-yloxy)-2-hydroxypropyl][2-(2-met...)
Affinity DataKd:  1.76nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2008
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKd:  1.80nMAssay Description:Antagonist activity at human beta-1 adrenergic receptor site 1 expressed in cimeterol-stimulated CHO-K1 cells assessed as CRE-SPAP level by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25748BDBM25748(ICI 89,406 | 3-(2-{[3-(2-cyanophenoxy)-2-hydroxypr...)
Affinity DataKd:  1.80nMAssay Description:Displacement of [3H]-CGP12177 from human beta1 adrenoceptor expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404994BDBM50404994(CHEMBL2096752)
Affinity DataKd:  1.90nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81886BDBM81886(CHEMBL287651 | CAS_3506-09-0 | PROPRANOLOL, dl)
Affinity DataKd:  2nMAssay Description:In vitro ability to block beta-1 adrenergic receptor in guinea pig right atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKd:  2nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404695BDBM50404695(CHEMBL174853)
Affinity DataKd:  2nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKd:  2.40nMAssay Description:Beta-1 adrenergic receptor blocking activity in atria of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKd:  2.40nMAssay Description:Antagonism of the isoprenaline-induced positive chronotropic effect on the atria of guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Regensburg

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019443BDBM50019443(LB-46 | 1-(1H-Indol-4-yloxy)-3-isopropylamino-prop...)
Affinity DataKd:  2.40nMAssay Description:Antagonist activity at human beta-1 adrenergic receptor site 1 expressed in cimeterol-stimulated CHO-K1 cells assessed as CRE-SPAP level by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
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