Compile Data Set for Download or QSAR
Report error Found 7 of kd data for polymerid = 3629,7888,11048,49000190,49000199,49000200,49000203
TargetAlpha-1B adrenergic receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50414756(CHEMBL569201)
Affinity DataKd:  281nMAssay Description:Antagonist activity at Alpha-1B adrenoceptor in guinea pig spleen assessed as inhibition of noradrenaline-induced contraction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKd:  0.676nMAssay Description:Antagonist activity at alpha1B adrenoceptor in Sprague-Dawley rat spleen assessed as inhibition of phenylephrine-induced contractions after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392639(CHEMBL2153551)
Affinity DataKd:  15.8nMAssay Description:Antagonist activity at alpha1B adrenoceptor in Sprague-Dawley rat spleen assessed as inhibition of phenylephrine-induced contractions after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392641(CHEMBL2153553)
Affinity DataKd:  0.263nMAssay Description:Antagonist activity at alpha1B adrenoceptor in Sprague-Dawley rat spleen assessed as inhibition of phenylephrine-induced contractions after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392643(CHEMBL2153555)
Affinity DataKd:  8.91nMAssay Description:Antagonist activity at alpha1B adrenoceptor in Sprague-Dawley rat spleen assessed as inhibition of phenylephrine-induced contractions after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392645(CHEMBL2153557)
Affinity DataKd:  2.75nMAssay Description:Antagonist activity at alpha1B adrenoceptor in Sprague-Dawley rat spleen assessed as inhibition of phenylephrine-induced contractions after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392647(CHEMBL2153559)
Affinity DataKd:  16.6nMAssay Description:Antagonist activity at alpha1B adrenoceptor in Sprague-Dawley rat spleen assessed as inhibition of phenylephrine-induced contractions after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed