Compile Data Set for Download or QSAR
Report error Found 29 of kd data for polymerid = 4341,49000160,50001766,50002434
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268107BDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKd:  0.170nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Mouse)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268232BDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKd:  0.351nMAssay Description:Displacement of [3H]PSB-603 from mouse recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268232BDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKd:  0.403nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cells by saturation experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268232BDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKd:  0.652nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cells by kinetic experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086170BDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataKd:  1.13nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229885BDBM50229885(N-(benzo[d][1,3]dioxol-5-yl)-2-(5-(2,6-dioxo-1,3-d...)
Affinity DataKd:  1.65nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229885BDBM50229885(N-(benzo[d][1,3]dioxol-5-yl)-2-(5-(2,6-dioxo-1,3-d...)
Affinity DataKd:  1.70nMAssay Description:Binding affinity of [3H]-MRE 2029-F20 towards human adenosine A2b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583640BDBM50583640(CHEMBL5075285)
Affinity DataKd:  7.80nMAssay Description:Binding affinity to NLuc human A2B adenosine receptor expressed in HEK293-A cells in presence of 1 uM PSB603 by NanoBRET binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026636BDBM50026636(RAUWOLSCINE HYDROCHLORIDE | 17alpha-hydroxy-20alph...)
Affinity DataKd:  13.8nMAssay Description:In vitro presynaptic agonist potency at alpha-2 adrenergic receptor in rat or mouse vas deferens relative to clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026636BDBM50026636(RAUWOLSCINE HYDROCHLORIDE | 17alpha-hydroxy-20alph...)
Affinity DataKd:  14nMAssay Description:In vitro presynaptic agonist potency at alpha-2 adrenergic receptor in rat or mouse vas deferens relative to clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583644BDBM50583644(CHEMBL5080679)
Affinity DataKd:  55nMAssay Description:Binding affinity to NLuc human A2B adenosine receptor expressed in HEK293-A cells in presence of 1 uM PSB603 by NanoBRET binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268085BDBM50268085(CHEMBL490262 | SB-298 | CHEMBL521280 | N-(2-hydrox...)
Affinity DataKd:  60nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275499BDBM50275499(2-(4-fluorophenyl)-3-(4-pyridinyl)pyrazolo-[1,5-a]...)
Affinity DataKd:  280nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583641BDBM50583641(CHEMBL5086197)
Affinity DataKd: <1.00E+3nMAssay Description:Binding affinity to NLuc human A2B adenosine receptor expressed in HEK293-A cells in presence of 1 uM PSB603 by NanoBRET binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150074BDBM50150074(2-Amino-4-(4-hydroxy-phenyl)-6-(1H-imidazol-2-ylme...)
Affinity DataKd:  3.07E+3nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595382BDBM50595382(CHEMBL5208068)
Affinity DataKd:  1.93E+4nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595372BDBM50595372(CHEMBL5195119)
Affinity DataKd:  2.20E+4nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 6659BDBM6659(1-phenyl-3-pyridin-2-ylurea | cid_221427 | N-Pheny...)
Affinity DataKd:  4.33E+4nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595381BDBM50595381(CHEMBL5184937)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595376BDBM50595376(CHEMBL47633)
Affinity DataKd:  6.07E+4nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595374BDBM50595374(CHEMBL5197070)
Affinity DataKd:  8.00E+4nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595380BDBM50595380(BENZOGUANAMINE)
Affinity DataKd:  1.07E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595371BDBM50595371(CHEMBL5193006)
Affinity DataKd:  1.08E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207720BDBM50207720(CHEMBL3954022)
Affinity DataKd:  1.20E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520329BDBM50520329(CHEMBL4550896)
Affinity DataKd:  1.23E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 152260BDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  1.40E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595378BDBM50595378(CHEMBL5204663)
Affinity DataKd:  1.48E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595379BDBM50595379(CHEMBL5193059)
Affinity DataKd:  1.96E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595375BDBM50595375(CHEMBL1573515)
Affinity DataKd:  1.99E+5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed