Compile Data Set for Download or QSAR
Report error Found 7 of kd data for polymerid = 4392,9136
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM50358204(CHEMBL1922094)
Affinity DataKd:  9.80E+3nMAssay Description:Binding affinity to DNAPK (unknown origin) by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2019
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to DNAPK (unknown origin) by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2019
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM50308135(PKI-587 | 1-(4-{[4-(Dimethylamino)piperidin-1-yl]c...)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to DNAPK (unknown origin) by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2019
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM50240973(CHEMBL4102855)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to DNAPK (unknown origin) by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2019
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM50240975(CHEMBL4084907)
Affinity DataKd:  1.60E+3nMAssay Description:Binding affinity to DNAPK (unknown origin) by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2019
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM50380363(CHEMBL2017974 | US10173995, Compound 1)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to DNAPK (unknown origin) by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2019
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Basel

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  288nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed