TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.356nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M4 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 2.40nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M4 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 5.40nMAssay Description:Potency of the compound assessed to inhibit cAMP levels in rat striatum, for blocking oxotremorine-M, in functional assay for Muscarinic acetylcholin...More data for this Ligand-Target Pair