Affinity DataKd: 3.94E+3nMAssay Description:Displacement of [3H]S-glutamate from rat GluR5 S1S2 ligand binding core expressed in Escherichia coli (DE3)More data for this Ligand-Target Pair
Affinity DataKd: 1.88E+3nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 209nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 7.31E+4nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 6.05E+4nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 5.94E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.09E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 4.91E+4nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 8.17E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.78E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.66E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 358nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 1.38E+3nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 102nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 209nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 23nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 55nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 9.25E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair