TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 38.2nMAssay Description:Binding affinity against MCF cells in the membrane preparation using radioligand binding assay.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 1.24E+4nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as dissociation constant by competitive binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 34.5nMAssay Description:Binding affinity to Sigma opioid receptor type 1 sites in guinea pig brain membranes at 0.1 uM of BNITMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 11.6nMAssay Description:Binding constant (Kd) for [3H]-DTG binding to Sigma opioid receptor type 1 of guinea pig brain membranes at 200 nM concentration of the compoundMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 13.6nMAssay Description:Binding constant (Kd) for [3H]DTG binding to Sigma opioid receptor type 1 of guinea pig brain membranes at 1 uM BNITMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 11.6nMAssay Description:Binding constant (Kd) for [3H]DTG binding to Sigma opioid receptor type 1 of guinea pig brain membranes at 5 uM BNITMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 7.20nMAssay Description:Displacement of [125I]N-IAC44 from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Displacement of [125I]N-IACoc from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKd: 2.90nMAssay Description:Binding affinity to guinea pig brain sigma1 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKd: 2.90nMAssay Description:Binding affinity to sigma1 receptor in Hartley guinea pig brain cortex membranes incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from recombinant sigma 1 receptor (unknown origin) expressed in baculovirus infected Sf9 cell membranes after 1.5...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from recombinant sigma 1 receptor (unknown origin) expressed in baculovirus infected Sf9 cell membranes after 1.5...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from recombinant sigma 1 receptor (unknown origin) expressed in baculovirus infected Sf9 cell membranes after 1.5...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from recombinant sigma 1 receptor (unknown origin) expressed in baculovirus infected Sf9 cell membranes after 1.5...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from recombinant sigma 1 receptor (unknown origin) expressed in baculovirus infected Sf9 cell membranes after 1.5...More data for this Ligand-Target Pair
Affinity DataKd: 239nMAssay Description:Displacement of [3H]pentazocine from sigma-1 opioid receptor in rat liver membranes after 1 hr by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair