Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of kd data for polymerid = 50000161
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50153520((S)-2-ethoxy-4-(2-(3-methyl-1-(2-(piperidin-1-yl)p...)
Affinity DataKd:  50nMAssay Description:Displacement of [3H]glibenclamide from COS-1 cells expressing Sulfonylurea receptor 1 (SUR-1)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50153521(2-Methoxy-4-{[(S)-3-methyl-1-(2-piperidin-1-yl-phe...)
Affinity DataKd:  83nMAssay Description:Displacement of [3H]glibenclamide from COS-1 cells expressing Sulfonylurea receptor 1 (SUR-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50153522(2-(2-Fluoro-ethoxy)-4-{[(S)-3-methyl-1-(2-piperidi...)
Affinity DataKd:  134nMAssay Description:Displacement of [3H]glibenclamide from COS-1 cells expressing Sulfonylurea receptor 1 (SUR-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50025847(CHEMBL3330879)
Affinity DataKd:  2.10nMAssay Description:Binding affinity to SUR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50025834(CHEMBL3330880)
Affinity DataKd:  0.380nMAssay Description:Binding affinity to SUR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed