Compile Data Set for Download or QSAR
Report error Found 8 of kd data for polymerid = 50000293,50000822
TargetDNA (cytosine-5)-methyltransferase 3A(Mouse)
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544058BDBM50544058(CHEMBL4640631)
Affinity DataKd:  900nMAssay Description:Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 15 uM using 30-mer duplex DNA (22 AT bp) as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Mouse)
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544058BDBM50544058(CHEMBL4640631)
Affinity DataKd:  900nMAssay Description:Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 5 uM using 30-mer duplex DNA (22 AT bp) as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Mouse)
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544058BDBM50544058(CHEMBL4640631)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 5 uM using 30-mer duplex DNA (17 AT bp) as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Mouse)
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544058BDBM50544058(CHEMBL4640631)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 30 uM using 30-mer duplex DNA (22 AT bp) as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Mouse)
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544058BDBM50544058(CHEMBL4640631)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 15 uM using 30-mer duplex DNA (17 AT bp) as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Mouse)
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544058BDBM50544058(CHEMBL4640631)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 30 uM using 30-mer duplex DNA (17 AT bp) as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of Toronto

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657830BDBM50657830(CHEMBL6146761)
Affinity DataKd:  4.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of Toronto

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657831BDBM50657831(CHEMBL6146700)
Affinity DataKd:  1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed