Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of kd data for polymerid = 50007095,5366
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50225514(CHEMBL160277)
Affinity DataKd:  1.00E+4nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50225512(CHEMBL157187)
Affinity DataKd:  320nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50225513(CHEMBL423055)
Affinity DataKd:  470nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) binding in SF-49 lymphoma cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed