TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne
Curated by ChEMBL
The University Of Melbourne
Curated by ChEMBL
Affinity DataKd: 0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne
Curated by ChEMBL
The University Of Melbourne
Curated by ChEMBL
Affinity DataKd: 0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne
Curated by ChEMBL
The University Of Melbourne
Curated by ChEMBL
Affinity DataKd: 0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+4nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) bindingMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne
Curated by ChEMBL
The University Of Melbourne
Curated by ChEMBL
Affinity DataKd: 0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) bindingMore data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) binding in SF-49 lymphoma cellMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
The University Of Melbourne
Curated by ChEMBL
The University Of Melbourne
Curated by ChEMBL
Affinity DataKd: 0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair