TargetType-1 angiotensin II receptor(Cavia porcellus)
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
Affinity DataKd: 15.8nMAssay Description:Antagonist activity at angiotensin AT1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 9.77nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 5.01nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.0501nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.0501nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.631nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataKd: 3.55nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.0912nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.0794nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 1.51nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataKd: 1.38nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataKd: 3.98nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 5.01nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit thoracic aortic ringsMore data for this Ligand-Target Pair
Affinity DataKd: 3.98nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit thoracic aortic ringsMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit thoracic aortic ringsMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.0813nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
Affinity DataKd: 1.51nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 0.117nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:In vitro binding affinity against Angiotensin II receptor in rabbit aorta ringsMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:In vitro binding affinity against Angiotensin II receptor in rabbit aorta ringsMore data for this Ligand-Target Pair
Affinity DataKd: 7.90nMAssay Description:In vitro binding affinity against Angiotensin II receptor in rabbit aorta ringsMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 0.930nMAssay Description:Binding affinity to human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 0.540nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 58nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 750nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
Affinity DataKd: 6.92nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
Affinity DataKd: 4.79nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
Affinity DataKd: 3.16nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
Affinity DataKd: 3.60nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 2.24E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 490nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 5.80nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 6.46E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 224nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 1.55E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 2.75E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair