Compile Data Set for Download or QSAR
maximum 50k data
Found 121 of kd data for polymerid = 5550,49000265,49000266,50002396,50004273,50004685
TargetType-1 angiotensin II receptor(Cavia porcellus)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50417811(CHEMBL1668010)
Affinity DataKd:  15.8nMAssay Description:Antagonist activity at angiotensin AT1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049207(2-Butyl-6-(1-methoxy-1-methyl-ethyl)-3-[2'-(1H-tet...)
Affinity DataKd:  9.77nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50003387(2-Ethyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKd:  5.01nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50047126(2-Ethyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKd:  0.0501nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataKd:  0.0501nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049200(2-Ethyl-5,7-dimethyl-3-[9-(1H-tetrazol-5-ylmethyl)...)
Affinity DataKd:  0.631nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049184(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKd:  3.55nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049212(4'-(2-Cyclopropyl-7-methyl-imidazo[4,5-b]pyridin-3...)
Affinity DataKd:  2nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049188(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKd:  0.0912nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50003154(2-{Propyl-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50417812(CHEMBL352257 | ME-3221)
Affinity DataKd:  1.51nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50281524(CHEMBL123713 | [3,3-Diethyl-5-oxo-1-[2'-(1H-tetraz...)
Affinity DataKd:  12.6nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50044355(2,5-Dibutyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataKd:  1.38nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50417813(CHEMBL340315)
Affinity DataKd:  3.98nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049205(CHEMBL48602 | RWJ-46458 | [4-Ethyl-4-methyl-6-oxo-...)
Affinity DataKd:  1nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50417814(CHEMBL1668002)
Affinity DataKd:  5.01nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit thoracic aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50209824(CHEMBL245444 | methyl 3-(4-(2-(1H-tetrazol-5-yl)-1...)
Affinity DataKd:  3.98nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit thoracic aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKd:  12.6nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit thoracic aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049191(CHEMBL341716 | LY-235656 | N-[1-(1-Carboxy-heptyl)...)
Affinity DataKd:  100nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50006909(2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKd:  0.0813nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049183(2,7-Diethyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataKd:  1.51nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50403230(A-81080 | CHEMBL49410)
Affinity DataKd:  0.117nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049205(CHEMBL48602 | RWJ-46458 | [4-Ethyl-4-methyl-6-oxo-...)
Affinity DataKd:  2.5nMAssay Description:In vitro binding affinity against Angiotensin II receptor in rabbit aorta ringsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50403236(CHEMBL123208)
Affinity DataKd:  10nMAssay Description:In vitro binding affinity against Angiotensin II receptor in rabbit aorta ringsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50280333(CHEMBL49207 | [4,4-Diethyl-6-oxo-1-[2'-(1H-tetrazo...)
Affinity DataKd:  7.90nMAssay Description:In vitro binding affinity against Angiotensin II receptor in rabbit aorta ringsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKd:  2nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50159215(CHEMBL3787375)
Affinity DataKd:  0.930nMAssay Description:Binding affinity to human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052104(CHEMBL410812 | Sar-Arg-Val-Tyr-Asp-His-Apt-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052103(CHEMBL217873 | Sar-Arg-Val-Tyr-Glu-His-Apt-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052105(CHEMBL405938 | Sar-Arg-Val-Tyr-Cys-His-Pen-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052106(CHEMBL406170 | Sar-Arg-Val-Tyr-Cys-His-Mpc-Phe)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052108(CHEMBL415025 | Sar-Arg-Val-Tyr-Hcy-His-Mpc-Phe)
Affinity DataKd:  20nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052101(2-({1-[2-{2-[2-{2-[5-Guanidino-2-(2-methylamino-ac...)
Affinity DataKd:  0.540nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052109(CHEMBL412864 | Sar-Arg-Val-Tyr-Cys-His-Mpt-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052102(CHEMBL414918 | Sar-Arg-Val-D-Tyr-Pro-His-Pro-Phe)
Affinity DataKd:  58nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052110(CHEMBL216678 | Sar-Arg-Val-Tyr-Hcy-His-Mpt-Phe)
Affinity DataKd:  750nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKd:  12.6nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50363826(CHEMBL1947129)
Affinity DataKd:  6.92nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50363828(CHEMBL1947131)
Affinity DataKd:  4.79nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50363833(CHEMBL1945010)
Affinity DataKd:  3.16nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408260(CHEMBL415157)
Affinity DataKd:  3.60nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408259(CHEMBL402669)
Affinity DataKd:  2.24E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50422224(CHEMBL406888)
Affinity DataKd:  490nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKd:  5.80nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408263(CHEMBL411624)
Affinity DataKd:  6.46E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408261(CHEMBL384349)
Affinity DataKd:  224nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50422225(CHEMBL408098)
Affinity DataKd:  1.55E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50422226(CHEMBL412717)
Affinity DataKd:  7.60nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50422227(CHEMBL405031)
Affinity DataKd:  2.75E+3nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408262(CHEMBL268804)
Affinity DataKd:  17nMAssay Description:Dissociation constant for [125 I] Ang binding to type 1 Angiotensin II receptorof bovine adrenocortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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