Compile Data Set for Download or QSAR
maximum 50k data
Found 16 of kd data for polymerid = 5868,49000197,6432
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKd:  0.324nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50601574(CHEMBL5201074)
Affinity DataKd:  0.25nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392641(CHEMBL2153553)
Affinity DataKd:  2.82nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392643(CHEMBL2153555)
Affinity DataKd:  0.912nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392645(CHEMBL2153557)
Affinity DataKd:  1.20nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392647(CHEMBL2153559)
Affinity DataKd:  39.8nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKd:  0.105nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392639(CHEMBL2153551)
Affinity DataKd:  166nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392641(CHEMBL2153553)
Affinity DataKd:  1.70nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392643(CHEMBL2153555)
Affinity DataKd:  0.275nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392645(CHEMBL2153557)
Affinity DataKd:  28.8nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392647(CHEMBL2153559)
Affinity DataKd:  53.7nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostatic vas deferans assessed as inhibition of noradrenaline-induced contractions...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50568740(CHEMBL4860528)
Affinity DataKd:  0.25nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50601551(CHEMBL5207281)
Affinity DataKd:  0.25nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50601567(CHEMBL5206565)
Affinity DataKd:  0.25nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50392639(CHEMBL2153551)
Affinity DataKd:  50.1nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat prostate assessed as inhibition of noradrenaline-induced contractions after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed