Compile Data Set for Download or QSAR
maximum 50k data
Found 17 of kd data for polymerid = 6680,49000608,49000609,50007536,50007660
TargetGlucocorticoid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016931(CHEBI:31677 | HYDROCORTISONE HEMISUCCINATE | Hydro...)
Affinity DataKd:  190nMAssay Description:Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50550126(3en3hg4wsw | CHEBI:8382 | Cortan | Cortancyl | Dec...)
Affinity DataKd:  29nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016932(CHEMBL3273976)
Affinity DataKd:  7nMAssay Description:Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016933(CHEMBL3273977)
Affinity DataKd:  430nMAssay Description:Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataKd:  19nMAssay Description:Binding affinity to glucocorticoid receptorMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataKd:  19nMAssay Description:Inhibition of glucocorticoid receptor (unknown origin)More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataKd:  2nMAssay Description:Binding affinity to GR (unknown origin)More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataKd:  15nMAssay Description:Binding affinity to GR (unknown origin)More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50550121(CHEMBL4787613)
Affinity DataKd:  2.20nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50550122(CHEMBL4754182)
Affinity DataKd:  138nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50550123(CHEMBL4755113)
Affinity DataKd:  883nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50550124(CHEMBL4764990)
Affinity DataKd:  32nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50381733(CHEMBL2022651)
Affinity DataKd:  2.20nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50550125(CHEMBL4759037)
Affinity DataKd:  9nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50381724(CHEMBL2022858)
Affinity DataKd:  2.60nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataKd:  2.80nMAssay Description:Induction of translocation of human glucocorticoid receptor expressed in HEK293T cells transduced with lentiviral vector expressing H2B-mCherry and G...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM13775((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataKd:  43nMAssay Description:Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair