Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of kd data for polymerid = 7093
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd:  1.93E+4nMAssay Description:Binding affinity to UHRF1 TTD (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd:  3.20E+4nMAssay Description:Binding affinity to UHRF1 Y188A/Y191A double mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd: >1.83E+5nMAssay Description:Binding affinity to UHRF1 F278A mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd: >1.11E+5nMAssay Description:Binding affinity to UHRF1 M224A mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50578341(CHEMBL4860378)
Affinity DataKd:  2.07E+4nMAssay Description:Binding affinity to UHRF1 TTD variant loop (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair