TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKd: 1.93E+4nMAssay Description:Binding affinity to UHRF1 TTD (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKd: 3.20E+4nMAssay Description:Binding affinity to UHRF1 Y188A/Y191A double mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKd: >1.83E+5nMAssay Description:Binding affinity to UHRF1 F278A mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKd: >1.11E+5nMAssay Description:Binding affinity to UHRF1 M224A mutant (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKd: 2.07E+4nMAssay Description:Binding affinity to UHRF1 TTD variant loop (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair