TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.04E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 2.56E+4nMAssay Description:Binding affinity to sensorchip-immobilized human His-tagged CFTR F508 deletion mutant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.47E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: >3.00E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: >3.00E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.10E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.77E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 6.60E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 6.10E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 5.90E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 3.57E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: >3.00E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.15E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 7.20E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 2.30E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.00E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 4.90E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 5.00E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 7.30E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 6.40E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 1.18E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 4.00E+4nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 9.66E+3nMAssay Description:To measure the direct binding of small molecules with CFTR, the interaction between small molecules and membrane fragments derived from HEK293 cells ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 20.2nMAssay Description:To measure the direct binding of small molecules with CFTR, the interaction between small molecules and membrane fragments derived from HEK293 cells ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 900nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells assessed as iodide influxMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 3.82E+4nMAssay Description:Binding affinity to His-tagged human CFTR-F508del mutant by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 8.93E+4nMAssay Description:Binding affinity to His-tagged human CFTR-F508del mutant by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 7.28E+4nMAssay Description:Binding affinity to His-tagged human CFTR-F508del mutant by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 4.78E+4nMAssay Description:Binding affinity to sensorchip-immobilized human His-tagged CFTR F508 deletion mutant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.89E+5nMAssay Description:Binding affinity to sensorchip-immobilized human His-tagged CFTR F508 deletion mutant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 1.75E+5nMAssay Description:Binding affinity to sensorchip-immobilized human His-tagged CFTR F508 deletion mutant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
National Research Council (Itb-Cnr)
Curated by ChEMBL
National Research Council (Itb-Cnr)
Curated by ChEMBL
Affinity DataKd: 6.58E+4nMAssay Description:Binding affinity to sensorchip-immobilized human His-tagged CFTR F508 deletion mutant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Rattus norvegicus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKd: 2.20E+5nMAssay Description:Kd (half effective concentration) of compound against CFTR (cystic fibrosis transmembrane conductance regulator) in rat was determinedMore data for this Ligand-Target Pair