TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.00370nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.00850nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.0150nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.0770nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Mixed-type inhibition of AChE in mouse cerebral cortex using acetylthiocholine iodide as substrate by double reciprocal Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Binding affinity to mouse AChEMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.720nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.800nM ΔG°: -51.4kJ/mole IC50: 2.40nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of mouse AChE assessed as inhibition constant using acetylthiocholine iodide as substrate measured every 2 mins by lineweaver-burk plot an...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of fetal bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Noncompetitive inhibition of Torpedo californica AChE using ATCh as substrate preincubated for 90 mins followed by substrate addition by potentiometr...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Competitive inhibition of Torpedo californica AChE using ATCh as substrate preincubated for 90 mins followed by substrate addition by potentiometric ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity tested against acetylcholinesterase in Torpedo californicaMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.5nM ΔG°: -47.2kJ/mole IC50: 16nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Binding affinity towards Acetylcholinesterase from fetal bovine serumMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Compound was evaluated for the binding affinity by displacing [3H]oxotremorine from mouse cerebral cortex tissue.More data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Mixed-type reversible inhibition of bovine acetylcholinesterase using S-acetylthiocholine as substrate incubated for 20 mins prior to substrate addit...More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding affinity to mouse AChEMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of fetal bovine serum AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 16.7nMAssay Description:Binding affinity towards Acetylcholinesterase from fetal bovine serumMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 17.5nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -44.2kJ/molepH: 7.0 T: 2°CAssay Description:Assays were conducted at 25 C in 20 mM sodium phosphate buffer (pH 7.0) and 0.01% bovine serum albumin unless otherwise noted. AChE concentrations we...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity tested against acetylcholinesterase in Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
Affinity DataKi: 19.6nM ΔG°: -43.6kJ/mole IC50: 52nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of bovine AChE at 30 nM using S-acetylthiocholine as as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair