Compile Data Set for Download or QSAR
Report error Found 122 of ki data for polymerid = 1554,50000448,50000635,50002720
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524390(CHEMBL4475619)
Affinity DataKi:  5.30nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  9.30nMAssay Description:Inhibition of Sprague-Dawley rat brain cytosolic Adk using [2-3H]adenosine incubated for 15 mins by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524393(CHEMBL4448092)
Affinity DataKi:  16nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  16nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  17nMAssay Description:Inhibition of rat brain ADK expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524387(CHEMBL4566815)
Affinity DataKi:  19nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524392(CHEMBL4475059)
Affinity DataKi:  19nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524388(CHEMBL4449169)
Affinity DataKi:  20nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524389(CHEMBL4525944)
Affinity DataKi:  21nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524394(CHEMBL4539148)
Affinity DataKi:  23nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524383(CHEMBL4442160)
Affinity DataKi:  26nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  26nMAssay Description:Inhibition of recombinant human Adk using [U-14C]adenosine by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524384(CHEMBL4458246)
Affinity DataKi:  28nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  30nMAssay Description:Inhibition of purified human adenosine kinase using varying levels of [3H]Ado as substrate in presence of adenosine deaminase inhibitor deoxycoformyc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524385(CHEMBL4463459)
Affinity DataKi:  33nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50368712(CHEMBL608051)
Affinity DataKi:  40nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524386(CHEMBL4474951)
Affinity DataKi:  48nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50524391(CHEMBL2042164)
Affinity DataKi:  120nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50368710(CHEMBL607761)
Affinity DataKi:  150nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50368709(CHEMBL607766)
Affinity DataKi:  160nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50368707(CHEMBL612205)
Affinity DataKi:  170nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50533828(CHEMBL4570031)
Affinity DataKi:  184nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  210nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Ra ATCC 25177 adenosine kinase using varying levels of [3H]Ado as substrate in presence of adenosine deam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50614446(CHEMBL5283680)
Affinity DataKi:  232nMAssay Description:Binding affinity to ADK (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50368708(CHEMBL611890)
Affinity DataKi:  300nMAssay Description:Inhibition of human placental adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524383(CHEMBL4442160)
Affinity DataKi:  410nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50413747(CHEMBL61741)
Affinity DataKi:  700nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50413740(CHEMBL61915)
Affinity DataKi:  900nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM23617(NBTI | Nitrobenzylthioinosine | CHEMBL418509 | (2R...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50366949(CHEMBL418496 | CHEMBL611841 | BDBM50413728)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50412070(CHEMBL59168)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50366950(CHEMBL292374 | BDBM50413729 | CHEMBL608593)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50412038(CHEMBL540448)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524385(CHEMBL4463459)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50366955(CHEMBL61387 | CHEMBL610357 | BDBM50413731)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50240561((2R,3R,4S,5R)-2-(6-(benzylthio)-9H-purin-9-yl)-5-(...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50413748(CHEMBL58072)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50413743(CHEMBL61524)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50413742(CHEMBL59195)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50100587(2-(6-Amino-5-nitro-pyrimidin-4-ylamino)-5-hydroxym...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of adenosine kinase from undialyzed W1-L2 lysate (0-50 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50413751(CHEMBL61773)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50412062(CHEMBL294755)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50533823(CHEMBL494210)
Affinity DataKi:  5.04E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524391(CHEMBL2042164)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of recombinant human adenosine kinase expressed in Escherichia coli BL21 (DE3) using adenosine as substrate in presence of ATP and PEP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50252013(4-[(4-Cyanobenzyl)thio]-7-(beta-D-ribofuranosyl)-7...)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity to purified Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50533825(CHEMBL4460819)
Affinity DataKi:  5.44E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50533832(CHEMBL4524434)
Affinity DataKi:  5.64E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50252067(4-[(4-Methoxybenzyl)thio]-7-(beta-D-ribofuranosyl)...)
Affinity DataKi:  5.80E+3nMAssay Description:Binding affinity to purified Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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