Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki data for polymerid = 1563,50000755,50001266
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298243((2E,6E)-8-(2-diazo-3,3,3-trifluoropropanoyloxy)-3,...)
Affinity DataKi:  200nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298245(4-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...)
Affinity DataKi:  480nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298242((E)-4-(3-benzoylbenzyloxy)-3-methylbut-2-enyl diph...)
Affinity DataKi:  610nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed