Compile Data Set for Download or QSAR
maximum 50k data
Found 77 of ki data for polymerid = 2433,4995,9934,9969,5860
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  0.150nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  8nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  8nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291023((2R,3R,4R,5S)-1-[(E)-3-(tert-Butyl-dimethyl-silany...)
Affinity DataKi:  10nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  17nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291030((2R,3R,4R,5S)-1-[4-(Dimethyl-phenyl-silanyl)-butyl...)
Affinity DataKi:  18nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM18353((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Affinity DataKi:  20nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  24nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  27nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  33nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291030((2R,3R,4R,5S)-1-[4-(Dimethyl-phenyl-silanyl)-butyl...)
Affinity DataKi:  39nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  40nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  50nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50242818(1-Oxo-1lambda-4-thia-cyclotridecan-3,4,5,6,8,10,11...)
Affinity DataKi:  52nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291032((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  55nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291027((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  64nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  100nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291028((2R,3R,4R,5S)-1-(Dimethyl-propyl-silanylmethyl)-2-...)
Affinity DataKi:  110nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  120nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291022((2R,3R,4R,5S)-2-Hydroxymethyl-1-trimethylsilanylme...)
Affinity DataKi:  150nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291033((2R,3R,4R,5S)-1-[(Dimethyl-phenyl-silanyl)-methyl]...)
Affinity DataKi:  160nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50147013(CHEMBL3764559)
Affinity DataKi:  185nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataKi:  200nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50147016(CHEMBL3763300)
Affinity DataKi:  210nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50147107(CHEMBL3763319)
Affinity DataKi:  216nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291025((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-4-trimethylsi...)
Affinity DataKi:  220nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291035((2R,3R,4R,5S)-2-Hydroxymethyl-1-((Z)-3-trimethylsi...)
Affinity DataKi:  350nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50147158(CHEMBL3764745)
Affinity DataKi:  353nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291023((2R,3R,4R,5S)-1-[(E)-3-(tert-Butyl-dimethyl-silany...)
Affinity DataKi:  390nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  420nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291035((2R,3R,4R,5S)-2-Hydroxymethyl-1-((Z)-3-trimethylsi...)
Affinity DataKi:  640nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50147159(CHEMBL3764813)
Affinity DataKi:  785nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291027((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  830nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84968(Urea derivative, 12)
Affinity DataKi:  3.20E+3nM IC50:  8.40E+3nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291022((2R,3R,4R,5S)-2-Hydroxymethyl-1-trimethylsilanylme...)
Affinity DataKi:  3.30E+3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291033((2R,3R,4R,5S)-1-[(Dimethyl-phenyl-silanyl)-methyl]...)
Affinity DataKi:  3.50E+3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291024((2R,3R,4R,5S)-2-Hydroxymethyl-1-(2-trimethylsilany...)
Affinity DataKi:  4.00E+3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50373981(CHEMBL403239)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of sucrose hydrolyzing activity of rat intestinal alpha glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50242818(1-Oxo-1lambda-4-thia-cyclotridecan-3,4,5,6,8,10,11...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84969(Urea derivative, 13)
Affinity DataKi:  4.60E+3nM IC50:  1.43E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Universidad Nacional Aut£Noma De M£Xico

Curated by ChEMBL
LigandPNGBDBM50341204((Z)-3-butylidenephthalide | CHEMBL1765390)
Affinity DataKi:  4.86E+3nMAssay Description:Mixed type inhibition of baker's yeast alpha-glucosidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291028((2R,3R,4R,5S)-1-(Dimethyl-propyl-silanylmethyl)-2-...)
Affinity DataKi:  7.00E+3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84967(Urea derivative, 11)
Affinity DataKi:  7.20E+3nM IC50:  1.98E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291024((2R,3R,4R,5S)-2-Hydroxymethyl-1-(2-trimethylsilany...)
Affinity DataKi:  8.50E+3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84972(Urea derivative, 16)
Affinity DataKi:  9.40E+3nM IC50:  1.85E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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