Compile Data Set for Download or QSAR
Report error Found 100 of ki data for polymerid = 3930,4170
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50210070(CHEMBL3883565)
Affinity DataKi: <0.100nMAssay Description:Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558851(CHEMBL4782684)
Affinity DataKi:  10nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558852(CHEMBL4747465)
Affinity DataKi:  31nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50210069(CHEMBL3884841)
Affinity DataKi:  32nMAssay Description:Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558857(CHEMBL4752520)
Affinity DataKi:  47nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558854(CHEMBL4755711)
Affinity DataKi:  82nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511123(CHEMBL4522193)
Affinity DataKi:  84nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511124(CHEMBL4533559)
Affinity DataKi:  100nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511138(CHEMBL4576854)
Affinity DataKi:  100nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511138(CHEMBL4576854)
Affinity DataKi:  100nMAssay Description:Displacement of fluorescent-labeled BID-BH3 peptide from His-tagged human BFL-1 (1 to 151 residues) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558856(CHEMBL4791348)
Affinity DataKi:  133nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511136(CHEMBL4558313)
Affinity DataKi:  150nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511125(CHEMBL4462138)
Affinity DataKi:  170nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558855(CHEMBL4740212)
Affinity DataKi:  175nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511139(CHEMBL4454113)
Affinity DataKi:  250nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511143(CHEMBL4463305)
Affinity DataKi:  280nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511122(CHEMBL4452560)
Affinity DataKi:  390nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM34194(3-chloro-1-(3,4-dichlorophenyl)-4-(4-methyl-1-pipe...)
Affinity DataKi:  400nMAssay Description:Displacement of fluorescent-labeled BID-BH3 peptide from His-tagged human BFL-1 (1 to 151 residues) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50604885(CHEMBL5177177)
Affinity DataKi:  410nMAssay Description:Displacement of fluorescein tagged BID BH3 peptide from His-tagged recombinant BFL-1 (1 to 151 residues) (unknown origin) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataKi:  430nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330257(6,6',7,7'-Tetrahydroxy-3,3'-dimethyl-5,5'-bis(2-ph...)
Affinity DataKi:  460nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM451097(US10676485, Example 7)
Affinity DataKi: >468nMAssay Description:Binding affinity to Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330256(5,5'-Bis(4-chlorobenzyl)-6,6',7,7''-tetrahydroxy-3...)
Affinity DataKi:  470nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330258(6,6',7,7'-Tetrahydroxy-3,3'-dimethyl-1,1',4,4'-tet...)
Affinity DataKi:  470nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511135(CHEMBL4457901)
Affinity DataKi:  570nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50621106(CHEMBL5401950)
Affinity DataKi:  630nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50078160(CHEMBL3417701)
Affinity DataKi: >660nMAssay Description:Inhibition of BCL2-A1 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511138(CHEMBL4576854)
Affinity DataKi:  680nMAssay Description:Displacement of fluorescein tagged BID BH3 peptide from His-tagged recombinant BFL-1 (1 to 151 residues) (unknown origin) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50621105(CHEMBL5420281)
Affinity DataKi:  750nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511137(CHEMBL4475729)
Affinity DataKi:  760nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511134(CHEMBL4435041)
Affinity DataKi:  810nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330251(N5,N5'-Bis(4-ethylphenethyl)-6,6',7,7'-tetrahydrox...)
Affinity DataKi:  870nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511144(CHEMBL4440719)
Affinity DataKi:  900nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330248(6,6',7,7'-Tetrahydroxy-5,5'-diisobutyl-3,3'-dimeth...)
Affinity DataKi:  930nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511146(CHEMBL4473975)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50376902(CHEMBL408194)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of BH3 peptide binding to human recombinant A1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50013888(CHEMBL3260038)
Affinity DataKi:  1.09E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511126(CHEMBL4525910)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50013865(CHEMBL3265297)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of Flu-BID/FAM-BID from His-tagged A1-BFL-1 (1 to 151) (unknown origin) expressed in Escherichia coli BL21(DE3) after 3 hrs by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50604880(CHEMBL5191993)
Affinity DataKi:  1.13E+3nMAssay Description:Displacement of fluorescein tagged BID BH3 peptide from His-tagged recombinant BFL-1 (1 to 151 residues) (unknown origin) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50635692(CHEMBL5527924)
Affinity DataKi:  1.27E+3nMAssay Description:Binding affinity to BFL-1 C55A mutant (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50635691(CHEMBL5523629)
Affinity DataKi:  1.38E+3nMAssay Description:Binding affinity to BFL-1 C55A mutant (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50621104(CHEMBL5440532)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330247(6,6',7,7'-Tetrahydroxy-5,5'-diisopropyl-3,3'-dimet...)
Affinity DataKi:  1.47E+3nMAssay Description:Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511128(CHEMBL4448621)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50621102(CHEMBL5438295)
Affinity DataKi:  1.63E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511145(CHEMBL4577267)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50621099(CHEMBL5413651)
Affinity DataKi:  1.84E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50621100(CHEMBL5418778)
Affinity DataKi:  1.92E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50635691(CHEMBL5523629)
Affinity DataKi:  1.95E+3nMAssay Description:Binding affinity to wild type human BFL-1 assessed as inhibition constant by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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