Compile Data Set for Download or QSAR
Report error Found 2 of ki data for polymerid = 4009
TargetBeta-secretase 1 [22-457](Human)
Philipps University Marburg

LigandPNGBDBM32389(phenyl-substituted sulfonamides, 6f)
Affinity DataKi:  6.40E+4nM ΔG°:  -23.9kJ/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1 [22-457](Human)
Philipps University Marburg

LigandPNGBDBM32386(phenyl-substituted sulfonamides, 6c)
Affinity DataKi:  1.50E+5nM ΔG°:  -21.8kJ/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed