Compile Data Set for Download or QSAR
Report error Found 3737 of ki data for polymerid = 4341,49000160,50001766,50002434
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511937(CHEMBL4552275)
Affinity DataKi:  0.0835nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Mouse)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511937(CHEMBL4552275)
Affinity DataKi:  0.131nMAssay Description:Displacement of [3H]PSB-603 from recombinant mouse A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511960(CHEMBL4450864)
Affinity DataKi:  0.137nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511968(CHEMBL4464522)
Affinity DataKi:  0.148nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511950(CHEMBL4540206)
Affinity DataKi:  0.153nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268151(1-Ethyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazin...)
Affinity DataKi:  0.157nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511961(CHEMBL4454481)
Affinity DataKi:  0.159nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50496142(CHEMBL3121728)
Affinity DataKi:  0.170nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cell membranes assessed as inhibition of NECA-stimulated adenylyl cycla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50455533(CHEMBL4205635)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine A2B receptor expressed in CHO cell membranes after 75 mins by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268109(8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phe...)
Affinity DataKi:  0.215nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511946(CHEMBL4463929)
Affinity DataKi:  0.215nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511973(CHEMBL4466625)
Affinity DataKi:  0.234nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511955(CHEMBL4567785)
Affinity DataKi:  0.244nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268164(1-Ethyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazin...)
Affinity DataKi:  0.281nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268163(1-Propyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazi...)
Affinity DataKi:  0.303nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511952(CHEMBL4460114)
Affinity DataKi:  0.342nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511964(CHEMBL4530074)
Affinity DataKi:  0.352nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268129(8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phe...)
Affinity DataKi:  0.393nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511948(CHEMBL4440526)
Affinity DataKi:  0.397nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50331916((S)-2-(2-oxo-4-phenethyl-3-(thiazol-2-yl)-1,2-dihy...)
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at adenosien A2B receptor in human HMC-1 cells assessed as inhibition of NECA-induced IL-8 release after 6 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM618748(US20230293517, Example 4.26)
Affinity DataKi:  0.400nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1×LabMed (Cisbio, France...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511959(CHEMBL4441276)
Affinity DataKi:  0.403nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268231(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.406nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511947(CHEMBL4454417)
Affinity DataKi:  0.421nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511940(CHEMBL4443090)
Affinity DataKi:  0.432nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50331917((R)-N-(2-hydroxy-1-phenylethyl)-2-(2-oxo-4-pheneth...)
Affinity DataKi:  0.440nMAssay Description:Antagonist activity at adenosien A2B receptor in human HMC-1 cells assessed as inhibition of NECA-induced IL-8 release after 6 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268150(8-(4-(4-(3-Fluorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.446nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50511957(CHEMBL4566170)
Affinity DataKi:  0.473nMAssay Description:Displacement of [3H]PSB-603 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins in presence of adeno...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268233(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.473nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM761402(N-[4-(3-Cyanophenyl)-5-(4-methyl-6-quinolyl)thiazo...)
Affinity DataKi:  0.5nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1× LabMed (Cisbio, Franc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to human recombinant A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50159502(CHEMBL3786849)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]OSIP339391 from human recombinant Adenosine A2B receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to human recombinant A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM761355(N-[4-(3-Cyanophenyl)-5-(1H-pyrrolo[2,3-b]pyridin-4...)
Affinity DataKi:  0.5nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1× LabMed (Cisbio, Franc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM761398(US20250243194, Example 7.29)
Affinity DataKi:  0.5nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1× LabMed (Cisbio, Franc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50159502(CHEMBL3786849)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]OSIP339391 from human recombinant adenosine A2B receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM761417(N-[4-(3-Cyanophenyl)-5-imidazo[1,2-a]pyridin-6-yl-...)
Affinity DataKi:  0.5nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1× LabMed (Cisbio, Franc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at human A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM761416(N-[4-(3-Cyanophenyl)-5-(3-methylbenzimidazol-5-yl)...)
Affinity DataKi:  0.5nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1× LabMed (Cisbio, Franc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM761424(N-[4-(3-Cyanophenyl)-5-pyrazolo[1,5-a]pyridin-5-yl...)
Affinity DataKi:  0.5nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1× LabMed (Cisbio, Franc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/12/2025
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268107(CHEMBL485862 | CHEMBL500634 | N-(2-(2-phenyl-6-(4-...)
Affinity DataKi:  0.5nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.553nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50268132(8-(4-(4-(4-Fluorobenzyl)piperazine-1-sulfonyl)phen...)
Affinity DataKi:  0.595nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM618723(US20230293517, Example 4.1 | 4-Cyano-N-[4-(3-cyano...)
Affinity DataKi:  0.600nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1×LabMed (Cisbio, France...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM618838(US20230293517, Example 6.68)
Affinity DataKi:  0.600nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1×LabMed (Cisbio, France...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM618870(US20230293517, Example 6.100)
Affinity DataKi:  0.600nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1×LabMed (Cisbio, France...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM618836(US20230293517, Example 6.66)
Affinity DataKi:  0.600nMAssay Description:All FRET binding experiments were conducted at room temperature in white 384-well plates, in assay binding buffer containing 1×LabMed (Cisbio, France...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Rheinische Friedrich-Wilhelms-Universitat Bonn

Curated by ChEMBL
LigandPNGBDBM50336996(N-[6-(2-Fluorophenyl)-5-(3-fluoropyridin-4-yl)pyra...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
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