Compile Data Set for Download or QSAR
Report error Found 8 of ki data for polymerid = 50000060
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487234(CHEMBL1391421)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50251868({(2Z)-3-[(6-chloropyridin-3-yl)methyl]-1,3-thiazol...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  3nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50486223(CHEBI:39164 | acetamiprid)
Affinity DataKi:  7.20nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50472282(descyanothiacloprid)
Affinity DataKi:  130nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  290nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50078048(1-(6-Chloro-pyridin-3-ylmethyl)-imidazolidin-(2Z)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit beta-like 2(Fruit fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed