Compile Data Set for Download or QSAR
maximum 50k data
Found 34 of ki data for polymerid = 50002220
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50513781(CHEMBL4466351)
Affinity DataKi:  0.340nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50513784(CHEMBL4550494)
Affinity DataKi:  0.730nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598266(CHEMBL5203652)
Affinity DataKi:  1.20nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598279(CHEMBL5199103)
Affinity DataKi:  1.40nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598286(CHEMBL5198215)
Affinity DataKi:  1.5nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598284(CHEMBL5176455)
Affinity DataKi:  1.90nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598268(CHEMBL5177587)
Affinity DataKi:  2nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598282(CHEMBL5205331)
Affinity DataKi:  2.20nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50513785(CHEMBL4575658)
Affinity DataKi:  2.40nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598278(CHEMBL5192991)
Affinity DataKi:  2.70nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598270(CHEMBL5203034)
Affinity DataKi:  2.70nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598283(CHEMBL5174330)
Affinity DataKi:  3.20nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598280(CHEMBL5175408)
Affinity DataKi:  3.60nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50513783(CHEMBL4456620)
Affinity DataKi:  3.70nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598281(CHEMBL5194536)
Affinity DataKi:  5.10nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598273(CHEMBL5194019)
Affinity DataKi:  5.80nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598269(CHEMBL5209454)
Affinity DataKi:  6.10nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598274(CHEMBL5172150)
Affinity DataKi:  6.40nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598267(CHEMBL5192120)
Affinity DataKi:  7nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50513782(CHEMBL4513520)
Affinity DataKi:  8.90nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598276(CHEMBL5181364)
Affinity DataKi:  11nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598265(CHEMBL5172861)
Affinity DataKi:  23nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598272(CHEMBL5196523)
Affinity DataKi:  24nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598271(CHEMBL5172332)
Affinity DataKi:  28nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598275(CHEMBL5203584)
Affinity DataKi:  29nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598277(CHEMBL5175074)
Affinity DataKi:  29nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50598285(CHEMBL5185690)
Affinity DataKi:  79nMAssay Description:Inhibition of C-terminal poly-His-tagged human recombinant KLK5 (30 to 293 residues) transfected in CHO cells assessed as inhibition constant using B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50513780(CHEMBL4456106)
Affinity DataKi:  143nMAssay Description:Inhibition of recombinant KLK5 (unknown origin) expressed in Pichia pastoris X-33 cells using pNA peptide as susbtrate measured every 10 secs for 300...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50256262(CHEMBL4070056)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human C-terminal 10His-tagged KLK5 (67 to 293 residues) expressed in mouse NS0 cells using fluorogenic Boc-VPR-AMC peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50507481(CHEMBL4564063)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris strain X-33 using Ac-YRSR-pNA as substrate preincubated for 30 mins followed by subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50507482(CHEMBL4531700)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris strain X-33 using Ac-YRSR-pNA as substrate preincubated for 30 mins followed by subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50507483(CHEMBL4530379)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris strain X-33 using Ac-YRSR-pNA as substrate preincubated for 30 mins followed by subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50256261(CHEMBL4059991)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of platelet-derived growth factor receptor beta phosphorylation in MG63 cells in the absence of plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50256260(CHEMBL4094403)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human C-terminal 10His-tagged KLK5 (67 to 293 residues) expressed in mouse NS0 cells using fluorogenic Boc-VPR-AMC peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed