Compile Data Set for Download or QSAR
maximum 50k data
Found 35 of ki data for polymerid = 50004321
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338966(CHEMBL1685065 | Phosphatidylinositol(3,4,5)-trisph...)
Affinity DataKi:  500nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338967(CHEMBL1685066 | D-3-deoxyphosphatidylinositol ethe...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50304369(4-dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonam...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338956(CHEMBL1685055 | Ethyl 2-(5-(4-Dodecylphenylsulfona...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338955(2-(5-(4-Dodecylphenylsulfonamido)-1,3,4-thiadiazol...)
Affinity DataKi:  5.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338949(4-Tetradecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfo...)
Affinity DataKi:  5.60E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338959(5-(4-Dodecylphenylsulfonamido)-1,3,4-thiadiazole-2...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338953(4-Dodecyl-N-(5-ethyl-1,3,4-thiadiazol-2-yl)benzene...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338958(4-Dodecyl-N-(5-(hydroxymethyl)-1,3,4-thiadiazol-2-...)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338950(4-Hexadecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfon...)
Affinity DataKi:  7.60E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338939(CHEMBL1685039 | N-(4-(N-(5-Ethyl-1,3,4-thiadiazol-...)
Affinity DataKi:  8.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338965(3-Dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonam...)
Affinity DataKi:  8.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338943(CHEMBL1685043 | Ethyl 5-(4-Decanamidophenylsulfona...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338942(CHEMBL1685042 | Ethyl 2-(5-(4-Decanamidophenylsulf...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338941(2-(5-(4-Decanamidophenylsulfonamido)-1,3,4-thiadia...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338938(CHEMBL1685038 | N-(4-(N-(5-Methyl-1,3,4-thiadiazol...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338944(CHEMBL1685044 | N-(4-(N-(5-(hydroxymethyl)-1,3,4-t...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338940(CHEMBL1685040 | N-(4-(N-(5-tert-Butyl-1,3,4-thiadi...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338951(4-Octadecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfon...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338961(CHEMBL1685060 | N-(5-Ethyl-1,3,4-thiadiazol-2-yl)b...)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338964(CHEMBL1685063 | ortho-Dodecyl-N-(1,3,4-thiadiazol-...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338960(CHEMBL1685059 | N-(1,3,4-Thiadiazol-2-yl)biphenyl-...)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338957(CHEMBL1685056 | Ethyl 5-(4-Dodecylphenylsulfonamid...)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50304368(CHEMBL595582 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338962(2-(5-(Biphen-4-ylsulfonamido)-1,3,4-thiadiazol-2-y...)
Affinity DataKi:  4.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50304371(CHEMBL611216 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50034417(4-Amino-N-[1,3,4]thiadiazol-2-yl-benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50304370(CHEMBL593946 | N-(4-(N-1,3,4-thiadiazol-2-ylsulfam...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338963(CHEMBL1685062 | para-Dodecyl-N-phenylbenzenesulfon...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338945(CHEMBL1685045 | N-(4-(N-(5-Sulfamoyl-1,3,4-thiadia...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338946(4-Butyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338947(4-Hexyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338952(4-Dodecyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzen...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338948(4-Octyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Mus musculus)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50338954(CHEMBL1685054 | N-(5-tert-Butyl-1,3,4-thiadiazol-2...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed