Compile Data Set for Download or QSAR
Report error Found 4 of ki data for polymerid = 50006125
TargetABC-type glutathione-S-conjugate transporter(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391002(CHEMBL2074599)
Affinity DataKi:  5.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetABC-type glutathione-S-conjugate transporter(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391003(CHEMBL493586)
Affinity DataKi:  1.05E+5nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetABC-type glutathione-S-conjugate transporter(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataKi:  3.37E+5nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetABC-type glutathione-S-conjugate transporter(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM18050(MTX | cid_126941 | Methotrexate | 2-[(4-{[(2,4-dia...)
Affinity DataKi:  1.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed