Compile Data Set for Download or QSAR
Report error Found 7 of ki data for polymerid = 50006845
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538688(CHEMBL4642789)
Affinity DataKi:  120nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50459608(CHEMBL3276621 | CHEBI:90441)
Affinity DataKi:  261nMAssay Description:Inhibition of human ALDH1A3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50585949(CHEMBL5083058)
Affinity DataKi:  460nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50527781(CHEMBL4456676)
Affinity DataKi:  540nMAssay Description:Competitive inhibition of recombinant human 6His-tagged ALDH1A3 expressed in Escherichia coli BL21(DE3) using varying level of acetaldehyde as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50585951(CHEMBL5086460)
Affinity DataKi: <1.00E+3nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50585950(CHEMBL5075900)
Affinity DataKi: <1.00E+3nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataKi:  8.70E+3nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed