Compile Data Set for Download or QSAR
Report error Found 13 of ki data for polymerid = 5138
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92449(Inhibitor, 19)
Affinity DataKi:  92nM ΔG°:  -40.2kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92445(US8691753, 105 | Inhibitor, 10)
Affinity DataKi:  113nM ΔG°:  -39.7kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92448(Inhibitor, 18)
Affinity DataKi:  406nM ΔG°:  -36.5kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92446(Inhibitor, 16)
Affinity DataKi:  1.26E+3nM ΔG°:  -33.7kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50183711(N-(4-(2-(hydroxyamino)-2-oxoethyl)piperidin-4-yl)-...)
Affinity DataKi:  1.83E+3nMAssay Description:Binding affinity to ADAMTS4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataKi:  2.68E+3nMAssay Description:Inhibition of ADAMTS-4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50183715(N-(4-(2-(hydroxyamino)-2-oxoethyl)tetrahydro-2H-py...)
Affinity DataKi:  4.60E+3nMAssay Description:Binding affinity to ADAMTS4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50183715(N-(4-(2-(hydroxyamino)-2-oxoethyl)tetrahydro-2H-py...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of ADAMTS4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50265114(N-((2R,6S)-4-(2-(hydroxyamino)-2-oxoethyl)-2,6-dim...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of ADAMTS4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50031472(CHEMBL307145 | 1,2,3-Trihydroxybenzene, XIV | pyro...)
Affinity DataKi:  6.34E+3nMAssay Description:Inhibition of ADAMTS-4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM26806((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)-1...)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of ADAMTS4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM92447(Inhibitor, 17)
Affinity DataKi: >1.00E+4nM ΔG°: >-28.5kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Human)
French Alternative Energies and Atomic Energy Commission

LigandPNGBDBM50305842(trans-4-((5-(2-(4-fluorobenzylcarbamoyl)-6-methylp...)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of ADAMTS4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed