Compile Data Set for Download or QSAR
maximum 50k data
Found 12 of ki data for polymerid = 5863,50003805,50006691,50006692,50006693
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50496737(CHEMBL3220783)
Affinity DataKi:  960nMAssay Description:Competitive inhibition of ThDP-dependent Escherichia coli DXP synthase using pyruvate as substrate assessed as NADPH consumption by spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Mycobacterium tuberculosis)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50026326(CHEMBL3305928)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis DXSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50496738(CHEMBL3220785)
Affinity DataKi:  5.60E+3nMAssay Description:Competitive inhibition of ThDP-dependent Escherichia coli DXP synthase using pyruvate as substrate assessed as NADPH consumption by spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli O127:H6 (strain E2348/69 / EPEC))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50026326(CHEMBL3305928)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of Escherichia coli DXSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli O127:H6 (strain E2348/69 / EPEC))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50026312(CHEMBL3306297)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of Escherichia coli DXSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50496736(CHEMBL3220784)
Affinity DataKi:  6.70E+3nMAssay Description:Competitive inhibition of ThDP-dependent Escherichia coli DXP synthase using pyruvate as substrate assessed as NADPH consumption by spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli O127:H6 (strain E2348/69 / EPEC))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50026348(CHEMBL3359030)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of Escherichia coli DXSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Haemophilus influenzae (strain 86-028NP))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50026349(KETOCLOMAZONE)
Affinity DataKi:  2.33E+4nMAssay Description:Inhibition of Haemophilus influenzae DXSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50496741(CHEMBL3220786)
Affinity DataKi:  2.58E+5nMAssay Description:Competitive inhibition of ThDP-dependent Escherichia coli DXP synthase using pyruvate as substrate assessed as NADPH consumption by spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM108228(1‐nitroso‐2‐naphthol (Substrate ...)
Affinity DataKi:  4.22E+5nM ΔG°:  -20.0kJ/mole IC50:  1.07E+6nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures containing HEPES (100mM, pH 8.0, 2mM MgCl2, 5mM NaCl), ThDP (1mM), BSA (1mg/mL), DMSO (10%, v/v), ᴅ-GAP (30µM), pyruvate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50496739(CHEMBL3220787)
Affinity DataKi: >1.00E+6nMAssay Description:Competitive inhibition of ThDP-dependent Escherichia coli DXP synthase using pyruvate as substrate assessed as NADPH consumption by spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose-5-phosphate synthase(Escherichia coli K-12 (Enterobacteria))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50496740(CHEMBL3220788)
Affinity DataKi: >1.00E+6nMAssay Description:Competitive inhibition of ThDP-dependent Escherichia coli DXP synthase using pyruvate as substrate assessed as NADPH consumption by spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed