Compile Data Set for Download or QSAR
Report error Found 95 of ki data for polymerid = 6170,49001148,50001613
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50530229(CHEMBL4460840)
Affinity DataKi:  0.120nMAssay Description:Inhibition of human CPB1 using AAFA as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50530229(CHEMBL4460840)
Affinity DataKi:  0.120nMAssay Description:Inhibition of human CPB1 using AAFA as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase B(Pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50201438((+/-)-5-guanidino-2-(mercaptomethyl)pentanoic acid...)
Affinity DataKi:  0.420nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305348((S)-2-(2-aminoethoxy)-3-(1-(2-cyclohexylethyl)-1H-...)
Affinity DataKi:  27nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305346((S)-2-(2-aminoethoxy)-3-(1-phenyl-1H-imidazol-4-yl...)
Affinity DataKi:  27nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305347((S)-2-(2-aminoethoxy)-3-(1-(4-tert-butylphenyl)-1H...)
Affinity DataKi:  49nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50226610((2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]...)
Affinity DataKi:  206nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50226610((2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]...)
Affinity DataKi:  206nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305345((S)-2-(2-aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl...)
Affinity DataKi:  238nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305352((S)-2-((R)-1-aminopropan-2-yloxy)-3-(1-phenyl-1H-i...)
Affinity DataKi:  240nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305351((S)-2-((R)-1-aminopropan-2-yloxy)-3-(1-(pyridin-2-...)
Affinity DataKi:  265nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305349((+/-)-2-(2-aminoethoxy)-3-(1-butyl-1H-imidazol-4-y...)
Affinity DataKi:  360nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM81910(1-((6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl...)
Affinity DataKi:  580nMAssay Description:The aromatic compounds screening were characterized by molecular docking as well as by in vitro inhibition assay against carboxypeptidase(CPs) of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296411(1-(4-chlorophenyl)-2-(5-(2-hydroxyphenyl)-1,3,4-ox...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270378(trans-1,1,3,3-tetraisopropyl-2-(3-(4-nitrophenyl)-...)
Affinity DataKi:  1.06E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296412(DL-guanidinoethylmercaptosuccinic acid | CHEMBL560...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50226606((S)-2-(2-aminoethylamino)-3-(1-propyl-1H-imidazol-...)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM81911(methyl 2-(3-furan-2-ylmethyl)-3-((8-methyl-2-oxo-1...)
Affinity DataKi:  1.20E+3nMAssay Description:The aromatic compounds screening were characterized by molecular docking as well as by in vitro inhibition assay against carboxypeptidase(CPs) of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296414(N-(3-chlorophenyl)-4-((5-(3-methoxybenzylthio)-1,3...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296413(N-benzyl-N-(4-phenylthiazol-2-yl)cyclopropanecarbo...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296415(4-(5-(2-chlorobenzylthio)-1,3,4-oxadiazol-2-yl)-N-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM81906(2-(5-(naphthalen-2-yloxy)methyl)-1,3,4-oxadiazol-2...)
Affinity DataKi:  1.60E+3nMAssay Description:The aromatic compounds screening were characterized by molecular docking as well as by in vitro inhibition assay against carboxypeptidase(CPs) of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305350((+/-)-2-(2-aminoethoxy)-3-(1-o-tolyl-1H-imidazol-4...)
Affinity DataKi:  2.72E+3nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270380(trans-1,1,3,3-tetraisopropyl-2-((2S,3S)-3-(4-metho...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296414(N-(3-chlorophenyl)-4-((5-(3-methoxybenzylthio)-1,3...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270379(trans-1,1,3,3-tetraisopropyl-2-((2S,3S)-3-(4-(trif...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM81905(1-(3,4-dihydroisoquinolin-1(1H)-yl)-2-(5-(3,5-dime...)
Affinity DataKi:  4.10E+3nMAssay Description:The aromatic compounds screening were characterized by molecular docking as well as by in vitro inhibition assay against carboxypeptidase(CPs) of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296413(N-benzyl-N-(4-phenylthiazol-2-yl)cyclopropanecarbo...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296416(methyl 2-(4-benzyl-5-(2-hydroxyphenyl)-4H-1,2,4-tr...)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50575780(CHEMBL4878039)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of recombinant human pancreatic CPB incubated for 25 mins using hippuryl-arginine as substrate by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270386(trans-(2RS,3RS)-3-(2-Thienyl)-2-trimethylsilyl-2-o...)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296417(isopropyl 2-(4-benzyl-5-(2-methoxyphenyl)-4H-1,2,4...)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296411(1-(4-chlorophenyl)-2-(5-(2-hydroxyphenyl)-1,3,4-ox...)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296418(2-(6,9-dimethyl-5H-[1,2,4]triazino[5,6-b]indol-3-y...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270381(trans-1,1,3,3-tetraisopropyl-2-((2S,3S)-3-p-tolyl-...)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM39191(cid_5447163 | 4-[4-(furan-2-ylmethyl)-3-(2-oxidany...)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270387(trans-(2RS,3RS)-3-(3-Thienyl)-2-trimethylsilyl-2-o...)
Affinity DataKi:  9.20E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50270385(trans-(2RS,3RS)-3-(4-Pyridyl)-2-trimethylsilyl-2-o...)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of human carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305353((+/-)-2-(2-(methylamino)ethoxy)-3-(1-propyl-1H-imi...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50305354((R)-2-(2-aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50121929(2-benzylbutanedioic acid | 2-benzylsuccinic acid |...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296420(ethyl 2-(4-ethyl-5-((4-ethylphenoxy)methyl)-4H-1,2...)
Affinity DataKi:  1.08E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296421(2-(4-benzyl-5-(thiophen-2-yl)-4H-1,2,4-triazol-3-y...)
Affinity DataKi:  1.16E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296422(2-(5-((4-chlorophenoxy)methyl)-1,3,4-oxadiazol-2-y...)
Affinity DataKi:  1.17E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296420(ethyl 2-(4-ethyl-5-((4-ethylphenoxy)methyl)-4H-1,2...)
Affinity DataKi:  1.19E+4nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50121929(2-benzylbutanedioic acid | 2-benzylsuccinic acid |...)
Affinity DataKi:  1.19E+4nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296422(2-(5-((4-chlorophenoxy)methyl)-1,3,4-oxadiazol-2-y...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM50296423(N-(2-chlorobenzyl)-N-(furan-2-ylmethyl)-3-methyl-4...)
Affinity DataKi:  1.26E+4nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCarboxypeptidase B(Corn earworm moth)
Universitat AutÒnoma De Barcelona

LigandPNGBDBM47512(SMR000003497 | 1-(4-methylphenyl)-2-[[5-(quinolin-...)
Affinity DataKi:  1.40E+4nMAssay Description:The aromatic compounds screening were characterized by molecular docking as well as by in vitro inhibition assay against carboxypeptidase(CPs) of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details Article
PubMed
TargetCarboxypeptidase B(Human)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296424(1-(2-fluorophenyl)-2-(5-o-tolyl-1,3,4-oxadiazol-2-...)
Affinity DataKi:  1.47E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
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