TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0300nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against adrenoceptor alpha 1AMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0700nMAssay Description:Inhibition of [3H]- prazosin binding against Alpha-1A adrenergic receptor from rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0800nMAssay Description:Overall binding displacement in tissues containing only the Alpha-1A adrenergic receptor from rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0900nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0900nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0900nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards alpha-1A adrenergic receptors using alpha1A ligand WB4101More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.210nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]prazosin from Alpha-1A adrenergic receptorof rat submaxillary gland membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.240nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.25nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]prazosin from Alpha-1A adrenergic receptorof rat submaxillary gland membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.270nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.270nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.270nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.280nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.290nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.320nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.330nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.330nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.350nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.360nMAssay Description:Binding affinity towards Alpha1A rat adrenergic receptors, using [125I]HEAT as radioligand.More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.380nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against adrenoceptor alpha 1AMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.390nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.410nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.430nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.440nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.480nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.490nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]prazosin from Alpha-1A adrenergic receptorof rat submaxillary gland membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair