Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of koff data for polymerid = 50000071,50001094,50001095,50000071,50001094,50001095
TargetProlyl endopeptidase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50279827(2-((S)-2-Formyl-pyrrolidine-1-carbonyl)-2,3-dihydr...)
Affinity DataKi:  2.40nM Kon:  0.000300M-1s-1 Koff:  1.40E+5s-1Assay Description:Compound was evaluated for the enzyme kinetic data (kon) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50279827(2-((S)-2-Formyl-pyrrolidine-1-carbonyl)-2,3-dihydr...)
Affinity DataKon:  0.000300M-1s-1Assay Description:Compound was evaluated for the enzyme kinetic data (koff) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50279826((1S,2S)-2-((S)-2-Formyl-pyrrolidine-1-carbonyl)-cy...)
Affinity DataKi:  3nM Kon:  0.000700M-1s-1 Koff:  2.30E+5s-1Assay Description:Compound was evaluated for the enzyme kinetic data (kon) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50279826((1S,2S)-2-((S)-2-Formyl-pyrrolidine-1-carbonyl)-cy...)
Affinity DataKon:  0.000700M-1s-1Assay Description:Compound was evaluated for the enzyme kinetic data (koff) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50279825((1R,2S)-2-((S)-2-Formyl-pyrrolidine-1-carbonyl)-cy...)
Affinity DataKi:  3nM Kon:  0.00200M-1s-1 Koff:  7.00E+5s-1Assay Description:Compound was evaluated for the enzyme kinetic data (kon) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50279825((1R,2S)-2-((S)-2-Formyl-pyrrolidine-1-carbonyl)-cy...)
Affinity DataKon:  0.00200M-1s-1Assay Description:Compound was evaluated for the enzyme kinetic data (koff) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article