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Found 1273 Enz. Inhib. hit(s) with Target = 'Chymotrypsin'
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(CHEMBL285285 | Peptide boronate)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(CHEMBL418050 | Peptide boronate)
Affinity DataKi:  0.0210nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(CHEMBL291026 | Peptide boronate)
Affinity DataKi:  0.115nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(CHEMBL290577 | Peptide boronate)
Affinity DataKi:  0.152nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(CHEMBL290577 | Peptide boronate)
Affinity DataKi:  0.365nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520048(CHEMBL4450993)
Affinity DataKi:  0.420nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014738(CHEMBL130253 | N-(Adamantyl-sulfonyl)-N-(methoxy s...)
Affinity DataKi:  0.580nMAssay Description:Binding affinity against human ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(CHEMBL2448441 | Peptide boronate)
Affinity DataKi:  0.848nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(CHEMBL2448441 | Peptide boronate)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520063(CHEMBL4586444)
Affinity DataKi:  0.880nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014735((1-{1-Methyl-2-oxo-2-[2-(3,3,3-trifluoro-1-isoprop...)
Affinity DataKi:  1nMAssay Description:Binding affinity against human ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034583(CHEMBL287918 | Peptide boronate)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034574(CHEMBL288150 | Peptide boronate)
Affinity DataKi:  1.21nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034576(CHEMBL288176 | Peptide boronate)
Affinity DataKi:  1.46nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520058(CHEMBL4469390)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034576(CHEMBL288176 | Peptide boronate)
Affinity DataKi:  2.20nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034573(CHEMBL291261 | Peptide boronate)
Affinity DataKi:  2.89nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034581(CHEMBL36744 | Peptide boronate)
Affinity DataKi:  2.96nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034574(CHEMBL288150 | Peptide boronate)
Affinity DataKi:  3.08nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataKi:  4.5nMAssay Description:Compound was evaluated for inactivation of bovine alpha-Chymotrypsin Kinetic constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(CHEMBL291026 | Peptide boronate)
Affinity DataKi:  4.56nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024092(6-Iodomethylene-4-phenyl-tetrahydro-pyran-2-one | ...)
Affinity DataKi:  5.30nMAssay Description:Binding constant of the compound alpha-chymotrypsin was determined by competitive inhibition assay with BTEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(CHEMBL285285 | Peptide boronate)
Affinity DataKi:  7.25nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(CHEMBL418050 | Peptide boronate)
Affinity DataKi:  8.08nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM87059(CHEMBL247767 | Chymostatin)
Affinity DataKi:  9.36nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM87059(CHEMBL247767 | Chymostatin)
Affinity DataKi:  9.36nMAssay Description:inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520064(CHEMBL4590739)
Affinity DataKi:  11nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50068892(3-(4-{[(S)-1-((S)-2-Acetylamino-3-methyl-butyryl)-...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for inhibitory activity against ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098882(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  12.6nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50061024((2-Methyl-1-{(S)-oxo-[(S)-2-((S)-3,3,3-trifluoro-1...)
Affinity DataKi:  13nMAssay Description:Binding affinity of the compound for porcine Pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50286327(4,6-Dimethoxy-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-...)
Affinity DataKi:  15nM Koff:  1.30E+3s-1Assay Description:Apparent binding constant Ki=Kon/KoffMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014738(CHEMBL130253 | N-(Adamantyl-sulfonyl)-N-(methoxy s...)
Affinity DataKi:  15nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50286327(4,6-Dimethoxy-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-...)
Affinity DataKi:  15nMAssay Description:Apparent binding constant Ki=Kon/KoffMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsinogen B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50014743(CHEMBL132171 | N-(1-{2-[2-(1-Benzyl-3,3,3-trifluor...)
Affinity DataKi:  17nMAssay Description:Binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50068901(3-[2,2-Difluoro-4-({(S)-1-[(S)-3-methyl-2-(3-pheny...)
Affinity DataKi:  19nMAssay Description:Compound was evaluated for inhibitory activity against ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50282866(4-Ethyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulf...)
Affinity DataKi:  20nM Koff:  1.30E+3s-1Assay Description:Apparent binding constant Ki=Kon/KoffMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)
Affinity DataKi:  20nMAssay Description:Inhibition of human chymotrypsin by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034581(CHEMBL36744 | Peptide boronate)
Affinity DataKi:  22.8nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50098842(2-(2-{2-[5-Amino-2-(4-fluoro-phenyl)-6-oxo-6H-pyri...)
Affinity DataKi:  23.3nMAssay Description:Inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50282868(1,1-Dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulfanylmeth...)
Affinity DataKi:  26nMAssay Description:Apparent binding constant Ki=Kon/KoffMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50282868(1,1-Dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulfanylmeth...)
Affinity DataKi:  26nM Koff:  130s-1Assay Description:Apparent binding constant Ki=Kon/KoffMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50031187(2-{(S)-2-[((S)-1-{(S)-2-[4-(4-Chloro-benzenesulfon...)
Affinity DataKi:  26nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014747(3-[(1-{2-[(1-Acetyl-pyrrolidine-2-carbonyl)-amino]...)
Affinity DataKi:  29nMAssay Description:Binding affinity against rat Cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014736((1-{1-Methyl-2-oxo-2-[2-(3,3,3-trifluoro-1-isoprop...)
Affinity DataKi:  32nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50098862(2-(2-{2-[5-Amino-2-(4-fluoro-phenyl)-6-oxo-6H-pyri...)
Affinity DataKi:  32.6nMAssay Description:Inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014730(CHEMBL130271 | N-(1-{1-Methyl-2-oxo-2-[2-(3,3,3-tr...)
Affinity DataKi:  33nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034583(CHEMBL287918 | Peptide boronate)
Affinity DataKi:  33.1nMAssay Description:Binding affinity of the compound towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068918((S)-4-((2S,3S)-2-Benzyloxycarbonylamino-3-methyl-p...)
Affinity DataKi:  34nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM247411(US10336754, Example 353 | US11053247, Example 353 ...)
Affinity DataKi:  35nMAssay Description:Binding affinity to human chymotrypsin assessed as inhibition constant using 3-Carbomethoxypropionyl-L-arginyl-Lprolyl-L-tyrosine p-Nitroaniline as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50282874(4-Isopropyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-yl...)
Affinity DataKi:  39nM Koff:  140s-1Assay Description:Apparent binding constant Ki=Kon/KoffMore data for this Ligand-Target Pair
In DepthDetails Article
Displayed 1 to 50 (of 1273 total ) | Next | Last >>
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