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Found 305 Enz. Inhib. hit(s) with Target = 'Pepsin A'
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012623(3-hydroxy-6-methyl-4-[2-methyl-1-[2-methyl-1-benzy...)
Affinity DataKi:  0nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012626(3-hydroxy-4-[2-methyl-1-[2-methyl-1-benzyloxycarbo...)
Affinity DataKi:  0nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataKi:  0nMAssay Description:Compound was measured for the inhibition of pepsin hydrolysis of hemoglobin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012624(3-hydroxy-4-[2-methyl-1-[2-methyl-1-benzyloxycarbo...)
Affinity DataKi:  0nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012622(3-hydroxy-4-[2-methyl-1-[2-methyl-1-benzyloxycarbo...)
Affinity DataKi:  0.0180nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012618(3-hydroxy-6-methyl-4-[2-methyl-1-[2-methyl-1-benzy...)
Affinity DataKi:  0.0390nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50028313(3-Hydroxy-6-methyl-4-{3-methyl-2-[3-methyl-2-(3-me...)
Affinity DataKi:  0.0457nMAssay Description:Pepsin inhibition was measured using the synthetic heptapeptide substrate Phe-Gly-His-Phe-(N02)-Phe-Ala- Phe-OMeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50141614((1S,2S,5S)-3-Hydroxy-4-[2-((S)-hydroxy-6-(S)-4-{(S...)
Affinity DataKi:  0.0460nMAssay Description:Inhibitory activity of the compound against aspartyl protease pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataKi:  0.0560nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50225475(CHEMBL92625)
Affinity DataKi: <0.100nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A-5(Homo sapiens (Human))
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50108795(CHEMBL3143435 | {1-[1-(1-{1-Hydroxy-1-methyl-2-[1-...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025532(3-Hydroxy-6-methyl-4-[3-methyl-2-(2-methyl-butyryl...)
Affinity DataKi:  0.180nMAssay Description:The compound was tested for inhibition of carboxyl protease (pepsin) inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025525(4-[2-(2-Ethyl-butyrylamino)-3-methyl-butyrylamino]...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested for inhibition of carboxyl protease (pepsin) inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012621(3-hydroxy-4-[2-methyl-1-[2-methyl-1-benzyloxycarbo...)
Affinity DataKi:  0.346nMAssay Description:Compound was measured for the apparent inhibition constant at pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025514(2-{2-[2-(4-{2-[2-(2-tert-Butoxycarbonylamino-3-phe...)
Affinity DataKi:  0.640nMAssay Description:Compound was tested for inhibition of pepsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50028314(CHEMBL325506 | N-(3-{1-Hydroxy-2-[1-(3-methyl-buty...)
Affinity DataKi:  0.900nMAssay Description:Pepsin inhibition was measured using the synthetic heptapeptide substrate Phe-Gly-His-Phe-(N02)-Phe-Ala- Phe-OMeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025899(3-Hydroxy-4-[3-methyl-2-(3-methyl-butyrylamino)-bu...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50022520(CHEMBL3349395 | H2N-Abu-Pro-Phe-Abu-Sta-Leu-PheOMe)
Affinity DataKi: <1nMpH: 4.0Assay Description:Inhibition of human renin at pH 6.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50227343(CHEMBL3349391)
Affinity DataKi: <1nMpH: 4.0Assay Description:Inhibition of porcine pepsin at pH 4.0 (time-dependent inhibition, T1/2>30 s)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50028312(3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  1.10nMAssay Description:Pepsin inhibition was measured using the synthetic heptapeptide substrate Phe-Gly-His-Phe-(N02)-Phe-Ala- Phe-OMeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50027905(3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  1.10nMAssay Description:Tested for time dependent inhibition constant against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012620(3-hydroxy-4-(4-hydroxyphenyl)-4-[2-methyl-1-[2-met...)
Affinity DataKi:  1.13nMAssay Description:Compound was measured for the inhibition of pepsin hydrolysis of hemoglobin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025889(3-Hydroxy-6-methyl-4-(methyl-{3-methyl-2-[3-methyl...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025889(3-Hydroxy-6-methyl-4-(methyl-{3-methyl-2-[3-methyl...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50027909(2-(2-{3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-b...)
Affinity DataKi:  1.5nMAssay Description:Tested for time dependent inhibition constant against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A-5(Homo sapiens (Human))
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50108798(CHEMBL3143437 | {1-[1-(1-{1-Hydroxy-2-[1-(3-methyl...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012619(3-hydroxy-4-(4-hydroxyphenyl)-4-[2-methyl-1-[2-met...)
Affinity DataKi:  1.54nMAssay Description:Compound was measured for the inhibition of pepsin hydrolysis of hemoglobin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025519(4-[2-(2,2-Dimethyl-propionylamino)-3-methyl-butyry...)
Affinity DataKi:  1.60nMAssay Description:The compound was tested for inhibition of carboxyl protease (pepsin) inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025510(2-{2-[2-(4-{2-[2-(2-tert-Butoxycarbonylamino-3-phe...)
Affinity DataKi:  1.70nMAssay Description:Compound was tested for inhibition of pepsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025901(4-Hydroxy-7-methyl-5-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50022293(CHEMBL124266 | N-(2-Hydroxy-1-isobutyl-4-{1-[1-(3-...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025513(2-[2-(4-{2-[2-(2-tert-Butoxycarbonylamino-3-phenyl...)
Affinity DataKi:  2.80nMAssay Description:Compound was tested for inhibition of pepsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50017485(1N-[1-isopentylcarbamoyl-(1S)-ethyl]-4-[1-(1-amino...)
Affinity DataKi:  2.90nMAssay Description:The compound was tested for inhibition of carboxyl protease (pepsin) inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50141612((S)-4-[(S)-2-(2-Amino-2-methyl-butyrylamino)-3-met...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity of the compound against aspartyl protease pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50022296(3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against porcine pepsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025890(4-Hydroxy-2,7-dimethyl-5-[3-methyl-2-(3-methyl-but...)
Affinity DataKi:  3nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025898(3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  3nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50027914(3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  3nMAssay Description:Tested for time dependent inhibition constant against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025890(4-Hydroxy-2,7-dimethyl-5-[3-methyl-2-(3-methyl-but...)
Affinity DataKi:  3nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50022305(CHEMBL123739 | N-{2-Hydroxy-1-isobutyl-4-[1-(2-iso...)
Affinity DataKi:  3nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50022302(CHEMBL339356 | N-(2-Hydroxy-1-isobutyl-4-{1-[1-(3-...)
Affinity DataKi:  3nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025526((1-{1-[1-(1-{1-Hydroxy-2-[1-(3-methyl-butylcarbamo...)
Affinity DataKi:  3.30nMAssay Description:Compound was tested for inhibition of pepsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025509(2-(3-Hydroxy-6-methyl-4-{3-methyl-2-[3-methyl-2-(3...)
Affinity DataKi:  3.5nMAssay Description:Tested for time dependent inhibition constant against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50022512(CHEMBL3349394 | Ibu-His-Pro-Phe-Ala-Sta-Leu-PheNH2)
Affinity DataKi:  4nMpH: 4.0Assay Description:Inhibition of porcine pepsin at pH 4.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50027915(3-Hydroxy-6-methyl-4-[3-methyl-2-(3-methyl-butyryl...)
Affinity DataKi:  4.60nMAssay Description:Tested for time dependent inhibition constant against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025528(2-[2-(4-{2-[2-(2-tert-Butoxycarbonylamino-3-phenyl...)
Affinity DataKi:  6.10nMAssay Description:Compound was tested for inhibition of pepsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50028392(4-[2-(3,3-Dimethyl-2-oxo-butylamino)-3-methyl-buty...)
Affinity DataKi:  7.5nMAssay Description:The compound was tested for inhibition of carboxyl protease (pepsin) inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025530(BDBM50028390 | CHEMBL166522 | [1-(1-{1-Hydroxy-2-[...)
Affinity DataKi:  8.60nMAssay Description:The compound was tested for inhibition of carboxyl protease (pepsin) inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025892(3-Hydroxy-6-methyl-4-{3-methyl-2-[3-methyl-2-(3-me...)
Affinity DataKi:  10nMAssay Description:Inhibition of porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50025517(3-Hydroxy-6-methyl-4-{3-methyl-2-[3-methyl-2-(3-me...)
Affinity DataKi:  10nMAssay Description:Tested for time independent inhibition constant against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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