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Found 4 Enz. Inhib. hit(s) with Target = 'Phosphatidylcholine-sterol acyltransferase'
TargetPhosphatidylcholine-sterol acyltransferase(Homo sapiens (Human))
Dalhousie University

LigandPNGBDBM92615(Difluoroketone phospholipid analogue, 3)
Affinity DataIC50:  28nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylcholine-sterol acyltransferase(Homo sapiens (Human))
Dalhousie University

LigandPNGBDBM92616(Difluoroketone phospholipid analogue, 4)
Affinity DataIC50:  60nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetPhosphatidylcholine-sterol acyltransferase(Homo sapiens (Human))
Dalhousie University

LigandPNGBDBM92614(Difluoroketone phospholipid analogue, 2)
Affinity DataIC50:  60nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylcholine-sterol acyltransferase(Homo sapiens (Human))
Dalhousie University

LigandPNGBDBM92613(Difluoroketone phospholipid analogue, 1)
Affinity DataIC50: >500nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails