TargetTubulin alpha chain-like 3/1A chain/1B chain/1C chain/3C chain/3E chain/4A chain/8 chain(Human)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of tubulin alpha in human A2780 cells assessed as reduction in cell growthMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 6.60E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 1.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 30 min by CD spectra analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.14E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.66E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Affinity DataIC50: 4.93E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 5.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 5.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 6.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 6.40E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 6.60E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 6.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 7.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 7.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 8.10E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 8.90E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 9.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University
The Ohio State University
Affinity DataIC50: 1.07E+5nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Affinity DataKd: 3.70E+3nMAssay Description:Binding affinity to Ovis aries (sheep) brain tubulin assessed as intrinsic tryptophan fluorescence after 30 min by fluorescence spectroscopic analysi...More data for this Ligand-Target Pair