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Found 30 Enz. Inhib. hit(s) with Target = 'Tubulin alpha chain'
LigandPNGBDBM50517652(CHEMBL4584084)
Affinity DataIC50:  540nMAssay Description:Inhibition of tubulin alpha in human A2780 cells assessed as reduction in cell growthMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Trypanosoma cruzi)
Howard University

US Patent
LigandPNGBDBM240700(US9422231, IMDNQ3)
Affinity DataIC50:  3.20E+3nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTubulin alpha chain(Trypanosoma cruzi)
Howard University

US Patent
LigandPNGBDBM50375664(CHEMBL404939 | US9422231, IMDNQ1)
Affinity DataIC50:  6.00E+3nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81744(Oryzalin Analogue, 3)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81745(Oryzalin Analogue, 4)
Affinity DataIC50:  6.60E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Trypanosoma cruzi)
Howard University

US Patent
LigandPNGBDBM240703(US9422231, IMDNQ10)
Affinity DataIC50:  8.00E+3nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTubulin alpha chain(Trypanosoma cruzi)
Howard University

US Patent
LigandPNGBDBM240701(US9422231, IMDNQ2)
Affinity DataIC50:  1.20E+4nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81746(Chembridge No 7992831, 5)
Affinity DataIC50:  1.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM50487731(CHEMBL2262117)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 30 min by CD spectra analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM50487731(CHEMBL2262117)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM86012(Chalcone, 11)
Affinity DataIC50:  2.03E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM50487732(CHEMBL2262305)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM50067040(((E,E)-1,7-bis(4-hydroxy-3-methoxyphenyl)-1,6-hept...)
Affinity DataIC50:  2.66E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha chain(Trypanosoma cruzi)
Howard University

US Patent
LigandPNGBDBM240702(US9422231, IMDNQ11)
Affinity DataIC50: >4.00E+4nMpH: 6.9 T: 2°CAssay Description:Tubulin assembly assays were conducted to assess tubulin polymerization inhibition. The assays were conducted in a 96-well microplate. Assembly react...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81743(Oryzalin, 1)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM86007(Chalcone, 6)
Affinity DataIC50:  4.93E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM50487733(CHEMBL2262116)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81747(Chembridge No 9067250, Class 1, 8)
Affinity DataIC50:  5.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81748(Chembridge No 7946770, Class 1, 9)
Affinity DataIC50:  5.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81753(Chembridge No 9035165, Class 2, 13)
Affinity DataIC50:  6.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81749(Chembridge No 7960631, Class 1, 10)
Affinity DataIC50:  6.40E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81752(Chembridge No 9035650, Class 2, 12)
Affinity DataIC50:  6.60E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81751(Chembridge No 9041709, Class 2, 11)
Affinity DataIC50:  6.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81750(Chembridge No 9063043, Class 1, 17)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81756(Chembridge No 9056942, Class 3, 7)
Affinity DataIC50:  7.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81758(Chembridge No 9044486, Class 4, 6)
Affinity DataIC50:  8.10E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81755(Chembridge No 9026860, Class 3, 14)
Affinity DataIC50:  8.90E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81754(Chembridge No 7944934, Class 2, 16)
Affinity DataIC50:  9.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81757(Chembridge No 9049411, Class 4, 15)
Affinity DataIC50:  1.07E+5nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Ovis aries)TBA
LigandPNGBDBM50487731(CHEMBL2262117)
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to Ovis aries (sheep) brain tubulin assessed as intrinsic tryptophan fluorescence after 30 min by fluorescence spectroscopic analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article