TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 1.30nMAssay Description:Binding affinity to human FRK using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: <10nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 17nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant PTK5 (218 to end residues) using GGEEEEYFELVKKKK as substrate incubated for 40 mins in presence of [gamma33P-ATP] by ...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 19nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 29nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 32nMAssay Description:Inhibition of human PTK5 in presence of ATP by radiometric assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 34nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 36nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant FrkMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 46nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant human PTK5 (218 to end residues) using GGEEEEYFELVKKKK as substrate incubated for 40 mins in presence of [gamma33P]ATP by s...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 52nMAssay Description:IC50 Table 13-20: The protocol calls for test compound of the invention to be incubated with kinase, substrate, cofactors, and radio-isotope-labeled ...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 53nMAssay Description:Inhibition of FRK (unknown origin) by TR-FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 55nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 55nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 62nMAssay Description:Inhibition of GST-tagged full length human recombinant FRK expressed in baculovirus using Fluorescein-Poly GT as substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 79nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate preincubated for 60 mins followed by [gamma-33P]-ATP addition and measured after 120 m...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 79nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate preincubated for 60 mins followed by [gamma-33P]-ATP addition and measured after 120 m...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 85nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 111nMAssay Description:Inhibition of human FRKMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 132nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 151nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 154nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 187nMAssay Description:Inhibition of human FRKMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 214nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 361nMAssay Description:Inhibition of human FRKMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 379nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate preincubated for 60 mins followed by [gamma-33P]-ATP addition and measured after 120 m...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 379nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate preincubated for 60 mins followed by [gamma-33P]-ATP addition and measured after 120 m...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 472nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 510nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged FRK (218 to end residues) expressed in baculovirus Sf21 insect cells preincubated for 5 mins f...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 530nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 550nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 550nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 550nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 550nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair