Report error Found 513 Enz. Inhib. hit(s) with Target = '3-oxoacyl-[acyl-carrier-protein] synthase 3'
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: 1.21E+5nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: 1.41E+5nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: 1.22E+3nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 0.610nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 1.49nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 1.99nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 2.84nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 3.09nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 3.53nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 3.53nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 3.61nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 3.76nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 4nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 8.47nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 28nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 28.1nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 31.4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 34nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 34.4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 50nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 56.0nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 56nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 62nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 62.1nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 95.9nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 96nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 110nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 110nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University
Curated by ChEMBL
Portland State University
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 160nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 160nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 160nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 160nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 220nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 220nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 240nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 240nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 250nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 250nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals
Quorex Pharmaceuticals
Affinity DataIC50: 270nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
