Compile Data Set for Download or QSAR
Report error Found 5949 Enz. Inhib. hit(s) with Target = '72 kDa type IV collagenase'
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50427868(CHEMBL2326366)
Affinity DataKd:  15nMAssay Description:Binding affinity to MMP-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541626(CHEMBL4646589)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to N-terminal (His6)-MBP tagged full-length human proMMP2 expressed in Escherichia coli BL21(DE3) RIL assessed as reduction in Rhod-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541627(CHEMBL4646183)
Affinity DataKd:  280nMAssay Description:Binding affinity to N-terminal (His6)-MBP tagged full-length human proMMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541626(CHEMBL4646589)
Affinity DataKd:  1nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541628(CHEMBL4635462)
Affinity DataKd:  7.40E+3nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541629(CHEMBL4633815)
Affinity DataKd:  6.30E+3nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541630(CHEMBL4633082)
Affinity DataKd:  2.20E+4nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541631(CHEMBL4633702)
Affinity DataKd:  2.10E+4nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541632(CHEMBL4642352)
Affinity DataKd:  2.10E+4nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541633(CHEMBL4645295)
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50541627(CHEMBL4646183)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to fluorescein-labeled D570-A583 epitope of human MMP2 expressed in Escherichia coli BL21(DE3) RIL incubated for 30 mins by FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM12074((2R)-2-{[4-(4-bromophenyl)benzene]sulfonamido}-3-m...)
Affinity DataIC50: 0.00400nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM11863(CHEMBL440498 | alpha-tetrahydropyran beta-sulfone ...)
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of APMA-activated recombinant human MMP-2 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2019
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM11863(CHEMBL440498 | alpha-tetrahydropyran beta-sulfone ...)
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of recombinant human AMPA-activated MMP2 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate measured after 40 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2018
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM11863(CHEMBL440498 | alpha-tetrahydropyran beta-sulfone ...)
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of human recombinant MMP2 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM11863(CHEMBL440498 | alpha-tetrahydropyran beta-sulfone ...)
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of human recombinant MMP2 using fluorescence peptide Cy3-PLGLK(Cy5Q)AR-NH2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50616392(CHEMBL5412341)
Affinity DataIC50: 0.0340nMAssay Description:Inhibition of human recombinant MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-N2 as substrate preincubated for 5 mins followed by substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM24025((2R)-3-methyl-2-[(4-phenylbenzene)sulfonamido]buta...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50175548(N-Hydroxy-2-(4-phenoxy-benzenesulfonylamino)-aceta...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Lys-Pro- Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 as substrate incubated for 2 hrs prior to substrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606383(CHEMBL5209489)
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50610465(CHEMBL5288452)
Affinity DataIC50: 0.0449nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606385(CHEMBL5203315)
Affinity DataIC50: 0.0460nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50082556(AG-3340 | 2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benz...)
Affinity DataIC50: 0.0480nMAssay Description:In vitro selective inhibition against matrix metalloprotease-2 (MMP-2) using fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50106026((S)-2,2-Dimethyl-4-[4-(pyridin-3-yloxy)-benzenesul...)
Affinity DataIC50: 0.0480nMAssay Description:Inhibitory concentration against Matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50523895(CHEMBL4522121)
Affinity DataIC50: 0.0480nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50592894(CHEMBL473539)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606395(CHEMBL5207094)
Affinity DataIC50: 0.0510nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606384(CHEMBL5183245)
Affinity DataIC50: 0.0550nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606386(CHEMBL5182207)
Affinity DataIC50: 0.0550nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50131941(2-(4'-Chloro-biphenyl-4-ylsulfanylmethyl)-N-hydrox...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibitory activity against matrix metalloprotease-2 (MMP2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50610466(CHEMBL5280430)
Affinity DataIC50: 0.0650nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606380(CHEMBL5191373)
Affinity DataIC50: 0.0660nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606390(CHEMBL5185612)
Affinity DataIC50: 0.0680nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50389101(CHEMBL2064548)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50137279(6-Hydroxy-2-(4-nitro-benzenesulfonyl)-1,2,3,4-tetr...)
Affinity DataIC50: 0.0760nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606381(CHEMBL5198135)
Affinity DataIC50: 0.0780nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606377(CHEMBL5186594)
Affinity DataIC50: 0.0830nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606378(CHEMBL5170274)
Affinity DataIC50: 0.0890nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50161330((R)-2-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-N-h...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50082556(AG-3340 | 2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benz...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606388(CHEMBL5203492)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50523894(CHEMBL4535400)
Affinity DataIC50: 0.0960nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50606382(CHEMBL5191820)
Affinity DataIC50: 0.0970nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50108135(2-(Formyl-hydroxy-amino)-3-[4-(4-trifluoromethoxy-...)
Affinity DataIC50: 0.0980nMAssay Description:In vitro selective inhibition against matrix metalloprotease-2 (MMP-2) using fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50071267((7S,8R,11S)-9-Oxo-8-[2-(4-propyl-phenyl)-ethyl]-2-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of fibroblast gelatinase A (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50343077(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(trifluoromet...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50096646(2-(4'-Chloro-biphenyl-4-yloxymethyl)-N-hydroxy-4-(...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50343077(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(trifluoromet...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human MMP2 assessed as cleavage of fluorogenic peptide MCAPro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50348652(CHEMBL1801429)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human MMP2 assessed as cleavage of fluorogenic peptide MCAPro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50348651(CHEMBL1801430)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human MMP2 assessed as cleavage of fluorogenic peptide MCAPro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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