Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1/A2a/A2b/A3'
TargetAdenosine receptor A1/A2a/A2b/A3(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282636(CHEMBL4163380)
Affinity DataEC50:  8.71E+3nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1/A2a/A2b/A3(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataEC50:  6.76E+4nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1/A2a/A2b/A3(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282640(CHEMBL4168653)
Affinity DataEC50:  5.13E+3nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1/A2a/A2b/A3(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282637(CHEMBL4167064)
Affinity DataEC50:  6.17E+4nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]CHA from rat brain adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224560(CHEMBL605654)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]CHA from rat brain adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataIC50: 95.7nMAssay Description:Displacement of [3H]CHA from rat brain adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataIC50: 96nMAssay Description:Displacement of [3H]CHA from rat brain adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224562(CHEMBL605067)
Affinity DataIC50: 2.02E+4nMAssay Description:Displacement of [3H]CHA from rat brain adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224561(CHEMBL605655)
Affinity DataIC50: 7.65E+4nMAssay Description:Displacement of [3H]CHA from rat brain adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  0.600nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016450(CHEMBL39503 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1,...)
Affinity DataKi:  1.20nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataKi:  1.30nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine in rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  1.40nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat testesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataKi:  1.40nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat testesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataKi:  1.60nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine in rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  1.60nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016451(CHEMBL37306 | N-[2-(2-Amino-acetylamino)-ethyl]-2-...)
Affinity DataKi:  2.10nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226936(CHEMBL37351)
Affinity DataKi:  4.30nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  5nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat fatMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataKi:  5.5nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataKi:  7nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat fatMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataKi:  9nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat fatMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataKi:  10nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  15nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50367589(CHEMBL611126 | CHEMBL3144091)
Affinity DataKi:  16nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50367270(CHEMBL606297)
Affinity DataKi:  16nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  23nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226935(CHEMBL3143947)
Affinity DataKi:  30nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226934(CHEMBL3143946)
Affinity DataKi:  35nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  50nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat fatMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  110nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat testesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  125nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50367267(CHEMBL605246)
Affinity DataKi:  210nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  500nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKi:  800nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  900nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataKi:  920nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  2.00E+3nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKi:  2.00E+3nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKi:  3.00E+3nMAssay Description:Antagonist binding of rN6-cyclohexyl-[3H]adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  4.50E+3nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  4.50E+3nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKi:  5.00E+3nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKi:  5.00E+3nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  9.00E+3nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10849(CHEMBL113 | 1,3,7-trimethyl-3,7-dihydropurine-2,6-...)
Affinity DataKi:  1.50E+4nMAssay Description:Antagonist binding of 2-chloro-[3H]-adenosine to rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  2.00E+4nMAssay Description:Antagonist binding of N6-cyclohexyl-[3H]-adenosine to rat testesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKi:  2.00E+4nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat fatMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  2.20E+4nMAssay Description:Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat fatMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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