Compile Data Set for Download or QSAR
Report error Found 1468 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b'
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406506(CHEMBL606305)
Affinity DataEC50:  3.80nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406509(CHEMBL605667)
Affinity DataEC50:  3.70nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50368543(CHEMBL605668)
Affinity DataEC50:  0.191nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406511(CHEMBL604836)
Affinity DataEC50:  1.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406507(CHEMBL604837)
Affinity DataEC50:  5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406498(CHEMBL605672)
Affinity DataEC50:  417nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406514(CHEMBL605873)
Affinity DataEC50:  3nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50406516(CHEMBL605048)
Affinity DataEC50:  22nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50453224(CHEMBL410873 | 2-(l-hexyn-l-yl)-adenosine-5'-N-met...)
Affinity DataEC50:  105nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50368347(CHEMBL610655)
Affinity DataEC50:  388nMAssay Description:Maximal NECA stimulation of adenylate cyclase via A2 receptors in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataEC50:  720nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452322(CHEMBL2093998)
Affinity DataEC50:  980nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367375(CHEMBL604834)
Affinity DataEC50:  1.55E+3nMAssay Description:Potency against human platelet A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367368(CHEMBL606290)
Affinity DataEC50:  3.40E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367377(CHEMBL606289)
Affinity DataEC50:  5.90E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367366(CHEMBL606288)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataEC50:  110nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367387(CHEMBL606503)
Affinity DataEC50:  950nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367364(CHEMBL603990)
Affinity DataEC50:  4.50E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452314(CHEMBL2094082)
Affinity DataEC50:  4.20E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367379(CHEMBL605239)
Affinity DataEC50:  6.40E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452316(CHEMBL2094084)
Affinity DataEC50:  340nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452317(CHEMBL2094085)
Affinity DataEC50:  820nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367380(CHEMBL605449)
Affinity DataEC50:  1.20E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367374(CHEMBL606285)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367386(CHEMBL603571)
Affinity DataEC50:  420nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452314(CHEMBL2094082)
Affinity DataEC50:  5.80E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452315(CHEMBL2094086)
Affinity DataEC50:  280nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367383(CHEMBL604207)
Affinity DataEC50:  1.68E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452315(CHEMBL2094086)
Affinity DataEC50:  260nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452317(CHEMBL2094085)
Affinity DataEC50:  750nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452316(CHEMBL2094084)
Affinity DataEC50:  470nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367369(CHEMBL605867)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367376(CHEMBL605866)
Affinity DataEC50:  5.70E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367383(CHEMBL604207)
Affinity DataEC50:  1.83E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367376(CHEMBL605866)
Affinity DataEC50:  1.56E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367369(CHEMBL605867)
Affinity DataEC50:  1.73E+4nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367367(CHEMBL603358)
Affinity DataEC50:  8.90E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50025446(CHEMBL604408)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452322(CHEMBL2093998)
Affinity DataEC50:  3.10E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452321(CHEMBL2093997)
Affinity DataEC50:  2.90E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452320(CHEMBL2093996)
Affinity DataEC50:  2.20E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50452318(CHEMBL2093995)
Affinity DataEC50:  2.37E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataEC50:  1.70E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50367380(CHEMBL605449)
Affinity DataEC50:  4.40E+3nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367368(CHEMBL606290)
Affinity DataEC50:  2.20E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367377(CHEMBL606289)
Affinity DataEC50:  6.30E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367366(CHEMBL606288)
Affinity DataEC50: >3.00E+4nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367375(CHEMBL604834)
Affinity DataEC50:  1.20E+3nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367384(CHEMBL606504)
Affinity DataEC50: >1.00E+5nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 1468 total ) | Next | Last >>
Jump to: