Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with Target = 'Amino acid transporter'
TargetAmino acid transporter heavy chain SLC3A2(Homo sapiens)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  5.33E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetAmino acid transporter heavy chain SLC3A2(Homo sapiens)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  347nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140134(CHEMBL3753869)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140131(CHEMBL3752249)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140083(CHEMBL3752210)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140127(CHEMBL3754498)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464408(US10793514, Compound 12)
Affinity DataIC50: 7.20E+3nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464426(US10793514, Compound 19)
Affinity DataIC50: 7.90E+3nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140081(CHEMBL3752103)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140133(CHEMBL3753592)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140122(CHEMBL3754053)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464424(US10793514, Compound 17)
Affinity DataIC50: 9.60E+3nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140129(CHEMBL3752700)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140082(CHEMBL3754059)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464405(US10793514, Compound 9)
Affinity DataIC50: 1.15E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464402(US10793514, Compound 6)
Affinity DataIC50: 1.19E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140125(CHEMBL3753808)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464427(US10793514, Compound 20)
Affinity DataIC50: 1.37E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140080(CHEMBL3754415)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464425(US10793514, Compound 18)
Affinity DataIC50: 1.75E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464430(US10793514, Compound 23)
Affinity DataIC50: 1.76E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140126(CHEMBL3752316)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140124(CHEMBL3754369)
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140079(CHEMBL3753404)
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140132(CHEMBL3752943)
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464417(US10793514, Compound 16)
Affinity DataIC50: 2.56E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464403(US10793514, Compound 7)
Affinity DataIC50: 2.60E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464414(US10793514, Compound 15)
Affinity DataIC50: 3.37E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464404(US10793514, Compound 8)
Affinity DataIC50: 3.38E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140130(CHEMBL3752483)
Affinity DataIC50: 3.63E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464409(US10793514, Compound 13)
Affinity DataIC50: 4.01E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140123(CHEMBL3753173)
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464428(US10793514, Compound 21)
Affinity DataIC50: 4.83E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464411(US10793514, Compound 14)
Affinity DataIC50: 5.08E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464401(US10793514, Compound 5)
Affinity DataIC50: 5.72E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464407(US10793514, Compound 11)
Affinity DataIC50: 5.96E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140128(CHEMBL3752494)
Affinity DataIC50: 6.82E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088537(CHEMBL6251 | US10189805, Compound 1)
Affinity DataIC50: 7.02E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140084(CHEMBL3753993)
Affinity DataIC50: 8.64E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464429(US10793514, Compound 22)
Affinity DataIC50: 8.91E+4nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM464406(US10793514, Compound 10)
Affinity DataIC50: 1.42E+5nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234288(CHEMBL4085113)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234283(CHEMBL4060165)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234285(CHEMBL4083894)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234284(CHEMBL4083473)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234291(CHEMBL4068819)
Affinity DataKi:  7.30E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234287(CHEMBL4100876)
Affinity DataKi:  7.70E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234280(CHEMBL4071517)
Affinity DataKi:  8.30E+4nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234279(CHEMBL4078902)
Affinity DataKi:  1.77E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetAmino acid transporter(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50234278(CHEMBL4103180)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of rat ASCT2 expressed in HEK293 cells assessed as inhibition of L-alanine/Na+ exchange by measuring reduction in SCN anion inward current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
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