Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Aromatase [1-48]'
TargetAromatase [1-48](Human)
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 18nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2012
Entry Details Article
PubMed
TargetAromatase [1-48](Human)
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85252(2,4-Trans-4'-hydroxy-4-imidazolyl-7-methoxyfla...)
Affinity DataIC50: 40nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2012
Entry Details Article
PubMed
TargetAromatase [1-48](Human)
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85253(2,4-Trans-4',7-dihydroxy-4-imidazolyl-7-methox...)
Affinity DataIC50: 77nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2012
Entry Details Article
PubMed
TargetAromatase [1-48](Human)
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85249(2,4-Trans-3'-hydroxy-4-imidazolyl-7-methoxyfla...)
Affinity DataIC50: 130nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2012
Entry Details Article
PubMed
TargetAromatase [1-48](Human)
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85251(2,4-Trans-4'-cyano-4-imidazolyl-7-methoxyflava...)
Affinity DataIC50: 133nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2012
Entry Details Article
PubMed
TargetAromatase [1-48](Human)
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85250(2,4-Trans-4'-chloro-4-imidazolyl-7-methoxyflav...)
Affinity DataIC50: 200nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2012
Entry Details Article
PubMed