Report error Found 1052 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor'
Affinity DataEC50: 480nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKd: 2.80E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 4.30E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 4.50E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cells; 0.2-16More data for this Ligand-Target Pair
Affinity DataKd: 1.01E+5nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 7.60E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 6.60E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 2.30E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 7.40E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 6.20E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 56nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKd: 1.58nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.0501nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.794nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.794nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.316nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 1.26nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.437nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.479nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.724nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.398nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
Affinity DataKd: 0.398nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
