Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with Target = 'Growth hormone-releasing hormone receptor'
LigandPNGBDBM50403630(L-162752 | CHEMBL558802)
Affinity DataEC50:  14nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403616(CHEMBL540805)
Affinity DataEC50:  2.30nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403617(CHEMBL552911)
Affinity DataEC50:  6.60nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403618(CHEMBL538004)
Affinity DataEC50:  1.30nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403619(CHEMBL545704)
Affinity DataEC50:  2.10nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403620(CHEMBL540001)
Affinity DataEC50:  10nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403621(CHEMBL553290)
Affinity DataEC50:  2.5nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403622(CHEMBL544769)
Affinity DataEC50:  2nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403623(CHEMBL540800)
Affinity DataEC50:  2.5nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403624(CHEMBL542653)
Affinity DataEC50:  1.5nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403625(CHEMBL545002)
Affinity DataEC50:  0.800nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403626(CHEMBL544536)
Affinity DataEC50:  2.90nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403627(CHEMBL545465)
Affinity DataEC50:  1nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403628(L-692585)
Affinity DataEC50:  3nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403629(CHEMBL553478)
Affinity DataEC50:  1.90nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403638(CHEMBL538008)
Affinity DataEC50:  1nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403632(CHEMBL558422)
Affinity DataEC50:  5.80nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403637(CHEMBL555821)
Affinity DataEC50:  8.30nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403633(CHEMBL554852)
Affinity DataEC50:  28nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403634(CHEMBL552657)
Affinity DataEC50:  7nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50049481(3-Amino-3-methyl-N-{2-oxo-1-[2'-(1H-tetrazol-5-yl)...)
Affinity DataEC50:  60nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403631(CHEMBL557206)
Affinity DataEC50:  17nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403635(CHEMBL553507)
Affinity DataEC50:  6nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50403636(CHEMBL545003)
Affinity DataEC50:  4.40nMAssay Description:Ability to release growth hormone in a rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGrowth hormone-releasing hormone receptor(Human)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM36351(CID148124 | Docetaxel)
Affinity DataIC50: 0.140nMAssay Description:Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004993(CHEMBL386366 | GRF-analogues)
Affinity DataIC50: 0.730nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004979(CHEMBL440262 | Tyr-Ala-Asp-Ala-Ile-Phe-Thr-Asn-Ser...)
Affinity DataIC50: 0.800nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004976(CHEMBL385308 | GRF-analogues)
Affinity DataIC50: 1.90nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004966(CHEMBL428135 | Tyr-Ala-Asp-Ala-Ile-Phe-Thr-D-Asn-S...)
Affinity DataIC50: 5.60nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004973(CHEMBL216479 | GRF-analogues)
Affinity DataIC50: 6.60nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004970(CHEMBL438545 | GRF-analogues)
Affinity DataIC50: 7.20nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004969(CHEMBL266658 | GRF-analogues)
Affinity DataIC50: 9.5nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004989(CHEMBL265167 | His-Ala-Asp-Ala-Ile-Phe-Thr-Ser-Ser...)
Affinity DataIC50: 9.80nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004978(CHEMBL262750 | GRF-analogues)
Affinity DataIC50: 14nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004992(CHEMBL427794 | GRF-analogues)
Affinity DataIC50: 17nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004974(CHEMBL413014 | Ac-hGRF(1-29)NH2 | Ac-Tyr-Ala-Asp-A...)
Affinity DataIC50: 18nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004994(CHEMBL437461 | GRF-analogues)
Affinity DataIC50: 20nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004985(CHEMBL414943 | GRF-analogues)
Affinity DataIC50: 20nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004968(CHEMBL439108 | GRF-analogues)
Affinity DataIC50: 22nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004972(CHEMBL427665 | GRF-analogues)
Affinity DataIC50: 44nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004980(CHEMBL262536 | GRF-analogues)
Affinity DataIC50: 45nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004971(CHEMBL412558 | GRF-analogues)
Affinity DataIC50: 95nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004981(CHEMBL264522 | GRF-analogues)
Affinity DataIC50: 120nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004991(CHEMBL411913 | GRF-analogues)
Affinity DataIC50: 130nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004988(CHEMBL269041 | GRF-analogues)
Affinity DataIC50: 217nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004990(CHEMBL428284 | GRF-analogues)
Affinity DataIC50: 311nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004962(CHEMBL439306 | GRF-analogues)
Affinity DataIC50: 377nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004984(CHEMBL415373 | GRF-analogues)
Affinity DataIC50: 836nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004963(CHEMBL428464 | GRF-analogues)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004964(CHEMBL412221 | GRF-analogues)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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