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Report error Found 22 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 4'
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50182597(5-acetyl-4,7-benzyloxy-6-hydroxybenzofuran | CHEMB...)
Affinity DataEC50: >2.00E+4nMAssay Description:Effect on blockade of Kv1.4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50182585(5-acetyl-7-(4'-bromo)benzyloxy-6-hydroxy-4-methoxy...)
Affinity DataEC50:  4.30E+3nMAssay Description:Effect on blockade of Kv1.4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50375409(CHEMBL408488)
Affinity DataEC50:  2.30E+3nMAssay Description:Inhibition of Kv1.4 channel inactivation expressed in xenopus oocytes by voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50375408(CHEMBL259345)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of Kv1.4 channel inactivation expressed in xenopus oocytes by voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50182587(5-acetyl-4-(4'-chloro)benzyloxy-6-hydroxy-7-methox...)
Affinity DataEC50:  4.80E+3nMAssay Description:Effect on blockade of Kv1.4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50279106(5-(4-phenoxybutoxy)psoralen | 4-(4-phenoxybutoxy)-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50: 230nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50: 380nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: 730nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50220547(oroidin base | oroidin | 4,5-Dibromo-1H-pyrrole-2-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50220547(oroidin base | oroidin | 4,5-Dibromo-1H-pyrrole-2-...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456970(CHEMBL3261431)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456977(CHEMBL3261430)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456971(CHEMBL4210636)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of Kv1.4 (unknown origin) expressed in HEK293 cells by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Institute of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50456973(Clathrodin)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed