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Report error Found 1212 Enz. Inhib. hit(s) with Target = 'Voltage-dependent N-type calcium channel subunit alpha-1B'
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295695(2-(3-aminopropoxy)-N-(4-(3-aminopropoxy)benzyl)-N-...)
Affinity DataEC50:  3.18E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295696(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  3.08E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295697(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  1.78E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295698(2-(3-Amino-propoxy)-N-(6-phenoxy-benzothiazol-2-yl...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295699(2-(3-Guanidino-propoxy)-N-(6-phenoxy-benzothiazol-...)
Affinity DataEC50:  3.30E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295700([4-(3-Amino-propoxy)-benzyl]-(6-phenoxy-benzothiaz...)
Affinity DataEC50:  7.60E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295701(N-(3-{4-[(6-Phenoxy-benzothiazol-2-ylamino)-methyl...)
Affinity DataEC50:  5.80E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295702([4-(3-Amino-propoxy)-benzyl]-(4-phenoxy-phenyl)-am...)
Affinity DataEC50:  3.40E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295703(2-(3-(4-((4-phenoxyphenylamino)methyl)phenoxy)prop...)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295704(3-{4-[(Benzhydryl-amino)-methyl]-phenoxy}-propylam...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295705(2-(3-(4-((benzhydrylamino)methyl)phenoxy)propyl)gu...)
Affinity DataEC50:  2.30E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295706(3-{4-[(2,2-Diphenyl-ethylamino)-methyl]-phenoxy}-p...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295707(2-(3-(4-((2,2-diphenylethylamino)methyl)phenoxy)pr...)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304180(2-(8-Aminooctanamido)-5-(3-aminopropoxy)-N-(4-phen...)
Affinity DataEC50:  7.20E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304181(5-(4-Aminobutoxy)-2-(6-aminohexanamido)-N-(4-pheno...)
Affinity DataEC50:  9.90E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304182(5-(4-Aminobutoxy)-2-(8-aminooctanamido)-N-(4-pheno...)
Affinity DataEC50:  9.00E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304183(2-(5-Guanidinopentanamido)-5-(3-guanidinopropoxy)-...)
Affinity DataEC50:  1.16E+5nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304184(2-(5-Guanidinohexanamido)-5-(3-guanidinopropoxy)-N...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304185(2-(5-Guanidino-octanamido)-5-(3-guanidinopropoxy)-...)
Affinity DataEC50:  1.30E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304186(2-(5-Guanidinohexanamido)-5-(3-guanidinobutoxy)-N-...)
Affinity DataEC50:  1.70E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304187(2-(5-Guanidino-octanamido)-5-(3-guanidinobutoxy)-N...)
Affinity DataEC50:  1.50E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304188(2-(8-Guanidinooctanamido)-5-(3-guanidinopropoxy)-N...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304189(N-(4-(4-Fluorophenoxy)phenyl)-2-(8-guanidinooctana...)
Affinity DataEC50:  6.00E+3nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304190(2-(5-Aminopentanamido)-5-(3-aminopropoxy)-N-(4-phe...)
Affinity DataEC50:  7.70E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304191(2-(6-Aminohexanamido)-5-(3-aminopropoxy)-N-(4-phen...)
Affinity DataEC50:  1.07E+5nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM10633(CHEMBL83980 | 3-{[6-(benzylamino)-9-(propan-2-yl)-...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM10636(6-(benzylamino)-2-[(2-hydroxyethyl)amino]-9-isopro...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM10909(R-2-[6-(Benzyl-methyl-amino)-9-isopropyl-9H-purin-...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400587(CHEMBL2206257)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400588(CHEMBL2206256)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50132003((Z)-1H,1''H-[2,3'']Biindolylidene-3,2''-dione 3-ox...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50366800(OLOMOUCINE II)
Affinity DataEC50:  8.00E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400563(CHEMBL2206241)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataEC50:  2.76E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400565(CHEMBL2206262)
Affinity DataEC50:  1.42E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400566(CHEMBL2206239)
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400564(CHEMBL2206242)
Affinity DataEC50:  7.21E+3nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50056163((S)-2-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamin...)
Affinity DataEC50:  5.70E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400567(CHEMBL2206248)
Affinity DataEC50: >7.00E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400568(CHEMBL2206240)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400569(CHEMBL2206255)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50378235(CHEMBL461557)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50358220(CHEMBL455389)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400570(CHEMBL2206254)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400571(CHEMBL2206253)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400572(CHEMBL2206252)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400573(CHEMBL2206251)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400574(CHEMBL2206250)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400575(CHEMBL2206249)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50400576(CHEMBL2206247)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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